Estrogenic activity of E2-conjugated GLP-1 is mediated by intracellular endolysosomal acidification and estrone metabolism.
E2 结合的 GLP-1 的雌激素活性是通过细胞内溶酶体酸化和雌酮代谢介导的
期刊:Molecular Metabolism
影响因子:6.6
doi:10.1016/j.molmet.2025.102136
Coupland Callum, Sun Na, Khalil Ahmed, Karaoglu Ãzüm Ezgi, Liskiewicz Arkadiusz, Liskiewicz Daniela, Grandl Gerald, Akindehin Seun, Maity Gandhari, Yang Bin, Finan Brian, Knerr Patrick, Douros Jonathan D, Walch Axel, DiMarchi Richard, Tschöp Matthias H, Müller Timo D, Novikoff Aaron