An allosteric cyclin E-CDK2 site mapped by paralog hopping with covalent probes.
利用共价探针通过旁系同源物跃迁定位变构细胞周期蛋白 E-CDK2 位点
期刊:Nature Chemical Biology
影响因子:13.7
doi:10.1038/s41589-024-01738-7
Zhang Yuanjin, Liu Zhonglin, Hirschi Marscha, Brodsky Oleg, Johnson Eric, Won Sang Joon, Nagata Asako, Bezwada Divya, Petroski Matthew D, Majmudar Jaimeen D, Niessen Sherry, VanArsdale Todd, Gilbert Adam M, Hayward Matthew M, Stewart Al E, Nager Andrew R, Melillo Bruno, Cravatt Benjamin F