日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Accuracy of Three-Dimensionally Printed, Patient-Specific Drill Guides for Implant Placement in Canine Cervical Vertebrae: A Cadaveric Study

三维打印患者特异性钻孔导板在犬颈椎种植体植入中的准确性:一项尸体研究

Ponticello, Christopher J; Mariani, Christopher L; Carrillo, Joshua M R; Zlotnick, Joshua A; Blodgett, Kristen Malinak; Gavitt, Ashley; Harrysson, Ola

Synthesis and Evaluation of Halogenated Pralidoximes in Reactivation of Organophosphate-Inhibited Cholinesterases

卤代碘解磷定在有机磷酸酯抑制的胆碱酯酶再活化中的合成与评价

Knittelova, Karolina; Prchalova, Eliska; Fuchsova, Adela; Andrys, Rudolf; Kohoutova, Zuzana; Rademacherova, Sara; Prchal, Lukas; Musilek, Kamil; Malinak, David

Cysteine conjugates of acetaminophen and p-aminophenol are potent inducers of cellular impairment in human proximal tubular kidney HK-2 cells

对乙酰氨基酚和对氨基苯酚的半胱氨酸结合物是人近端肾小管HK-2细胞损伤的强效诱导剂。

Rousar, Tomas; Handl, Jiri; Capek, Jan; Nyvltova, Pavlina; Rousarova, Erika; Kubat, Miroslav; Smid, Lenka; Vanova, Jana; Malinak, David; Musilek, Kamil; Cesla, Petr

Inhibitors of phosphoinositide 3-kinase (PI3K) and phosphoinositide 3-kinase-related protein kinase family (PIKK)

磷脂酰肌醇3-激酶(PI3K)和磷脂酰肌醇3-激酶相关蛋白激酶家族(PIKK)抑制剂

Huang, Xueqin; You, Li; Nepovimova, Eugenie; Psotka, Miroslav; Malinak, David; Valko, Marian; Sivak, Ladislav; Korabecny, Jan; Heger, Zbynek; Adam, Vojtech; Wu, Qinghua; Kuca, Kamil

STAT3 inhibitor Stattic and its analogues inhibit STAT3 phosphorylation and modulate cytokine secretion in senescent tumour cells

STAT3 抑制剂 Stattic 及其类似物可抑制 STAT3 磷酸化并调节衰老肿瘤细胞中的细胞因子分泌

Romana Mikyskova, Olena Sapega, Miroslav Psotka, Ondrej Novotny, Zdeněk Hodny, Sona Balintova, David Malinak, Jana Svobodova, Rudolf Andrys, David Rysanek, Kamil Musilek, Milan Reinis

Charged pyridinium oximes with thiocarboxamide moiety are equally or less effective reactivators of organophosphate-inhibited cholinesterases compared to analogous carboxamides

与类似的羧酰胺相比,带有硫代羧酰胺部分的带电吡啶肟对有机磷酸盐抑制的胆碱酯酶的再活化作用相同或更低

Zuzana Kohoutova, David Malinak, Rudolf Andrys, Jana Svobodova, Miroslav Psotka, Monika Schmidt, Lukas Prchal, Kamil Musilek

The Effect of Chemical Structure of OEG Ligand Shells with Quaternary Ammonium Moiety on the Colloidal Stabilization, Cellular Uptake and Photothermal Stability of Gold Nanorods

含季铵部分的OEG配体壳的化学结构对金纳米棒的胶体稳定性、细胞摄取和光热稳定性的影响

Sarka Salajkova, Filip Havel, Michal Sramek, Filip Novotny, David Malinak, Rafael Dolezal, Lukas Prchal, Marketa Benkova, Ondrej Soukup, Kamil Musilek, Kamil Kuca, Jiri Bartek, Jan Proska, Monika Zarska, Zdenek Hodny

Design, synthesis, and in vitro evaluation of BP-1-102 analogs with modified hydrophobic fragments for STAT3 inhibition

设计、合成并体外评估具有修饰疏水片段的 BP-1-102 类似物对 STAT3 的抑制作用

Patrik Oleksak, Miroslav Psotka, Marketa Vancurova, Olena Sapega, Jana Bieblova, Milan Reinis, David Rysanek, Romana Mikyskova, Katarina Chalupova, David Malinak, Jana Svobodova, Rudolf Andrys, Helena Rehulkova, Vojtech Skopek, Pham Ngoc Lam, Jiri Bartek, Zdenek Hodny, Kamil Musilek

Pyridinium-2-carbaldoximes with quinolinium carboxamide moiety are simultaneous reactivators of acetylcholinesterase and butyrylcholinesterase inhibited by nerve agent surrogates.

具有喹啉羧酰胺部分的吡啶-2-羧肟可同时复活被神经毒剂替代物抑制的乙酰胆碱酯酶和丁酰胆碱酯酶

Lee Hyun Myung, Andrys Rudolf, Jonczyk Jakub, Kim Kyuneun, Vishakantegowda Avinash G, Malinak David, Skarka Adam, Schmidt Monika, Vaskova Michaela, Latka Kamil, Bajda Marek, Jung Young-Sik, Malawska Barbara, Musilek Kamil

Synthesis, in vitro screening and molecular docking of isoquinolinium-5-carbaldoximes as acetylcholinesterase and butyrylcholinesterase reactivators

异喹啉-5-卡巴肟作为乙酰胆碱酯酶和丁酰胆碱酯酶活化剂的合成、体外筛选和分子对接

Malinak, David; Dolezal, Rafael; Hepnarova, Vendula; Hozova, Miroslava; Andrys, Rudolf; Bzonek, Petr; Racakova, Veronika; Korabecny, Jan; Gorecki, Lukas; Mezeiova, Eva; Psotka, Miroslav; Jun, Daniel; Kuca, Kamil; Musilek, Kamil