Indolequinone-Based Hypoxia-Activated Proteolysis Targeting Chimeras Selectively Degrade BRD4 in Hypoxic Cancer Cells
基于吲哚醌的缺氧激活蛋白水解靶向嵌合体选择性降解缺氧癌细胞中的BRD4
期刊:Journal of the American Chemical Society
影响因子:15.6
doi:10.1021/jacs.5c10240
Serafini, Marta; Twigger, Sophie A; Delfas, George; Mallerman, Maxim; Bailey, Elliot P; Calder, Ewen D D; Hammond, Ester M; Conway, Stuart J