日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Estimation of Dopamine D(1) Receptor Agonist Binding Kinetics Using Time-Resolved Functional Assays: Relation to Agonist-Induced Receptor Internalization by Investigational Antiparkinsonian Therapeutics.

利用时间分辨功能测定法估算多巴胺 D(1) 受体激动剂结合动力学:与研究性抗帕金森病疗法中激动剂诱导的受体内化的关系

Sahlholm Kristoffer, Svensson Peder, Malo Marcus, Andersson Daniel R, Betari Nibal

Development of 7TM receptor-ligand complex models using ligand-biased, semi-empirical helix-bundle repacking in torsion space: application to the agonist interaction of the human dopamine D2 receptor

利用配体偏向的半经验螺旋束重排方法在扭转空间构建7TM受体-配体复合物模型:应用于人多巴胺D2受体激动剂相互作用的研究

Malo, Marcus; Persson, Ronnie; Svensson, Peder; Luthman, Kristina; Brive, Lars

Investigation of D₂ receptor-agonist interactions using a combination of pharmacophore and receptor homology modeling

利用药效团和受体同源建模相结合的方法研究D₂受体激动剂相互作用

Malo, Marcus; Brive, Lars; Luthman, Kristina; Svensson, Peder

Investigation of D₁ receptor-agonist interactions and D₁/D₂ agonist selectivity using a combination of pharmacophore and receptor homology modeling

利用药效团和受体同源建模相结合的方法研究D₁受体激动剂相互作用和D₁/D₂激动剂选择性

Malo, Marcus; Brive, Lars; Luthman, Kristina; Svensson, Peder