日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Synthesis and Biological Evaluation of Tetrahydroisoquinoline Derivatives as Trypanocidal Agents

四氢异喹啉衍生物作为锥虫杀灭剂的合成及生物学评价

de Moura Lopes, João Paulo; Marques, Gabriel Vitor de Lima; Diniz, Lucas Abreu; Côrrea Santos, Viviane; Resende, Daniela de Melo; Murta, Silvane Maria Fonseca; Kohlhoff, Markus; Maltarollo, Vinícius Gonçalves; Ferreira, Rafaela Salgado; Oliveira, Renata Barbosa

Reading between the Chains: Surface Mapping and Druggable Pockets on the Biological Assemblies of DENV-2's Protein E

解读链间结构:登革病毒2型E蛋白生物组装体的表面映射和可成药口袋

Leite, Pedro T T F; Fernandes, Philipe O; Lacerda, Pedro S; Chagas, Marcelo A; Castilho, Marcelo S; Rocha, Willian R; Moraes, Adolfo Henrique; Maltarollo, Vinícius G

Bioactivity-Guided Isolation of β-Sitosterol From Terminalia glabrescens as a Potent Anti-Zika Virus Agent

从光叶榄仁树中生物活性导向分离β-谷甾醇作为强效抗寨卡病毒剂

Pereira, Rosângela Santos; Campana, Priscilla Rodrigues Valadares; Costa, Vivian Vasconcelos; Maltarollo, Vinícius Gonçalves; de Pádua, Rodrigo Maia; de Gomes, José Hugo Sousa; de Sousa, Grasiely Farias; de Souza Filho, José Dias; de Souza, Daniele da Glória; Teixeira, Mauro Martins; Braga, Fernão Castro

Discovery of benzyl carbamate inhibitors of coronavirus M(pro) enzymes from a legacy collection of cysteine protease inhibitors

从一系列已知的半胱氨酸蛋白酶抑制剂中发现冠状病毒M(pro)酶的苄基氨基甲酸酯抑制剂

Sá Magalhães Serafim, Mateus; Kronenberger, Thales; Francisco, Karol R; de Sousa Reis, Erik Vinicius; Gonçalves de Oliveira, Ellen; Marcelino E Oliveira, Fernanda Kelly; Serraglio Fortes, Isadora; Maciel Fernandes, Thaís Helena; Barbosa da Silva, Elany; Fajtova, Pavla; Skinner, Danielle E; Syed, Rafay O; Lage de Siqueira-Neto, Jair; Poso, Antti; Fernandes Mota, Bruno Eduardo; Alves Coelho-Dos-Reis, Jordana Grazziela; Santos Abrahão, Jônatas; Gonçalves Maltarollo, Vinícius; O'Donoghue, Anthony J; Caffrey, Conor R

Look What You Made Me Do: Discerning Feature for Classification of Endocrine-Disrupting Chemical Binding to Steroid Hormone Receptors

看看你都让我做了什么:内分泌干扰化学物质与类固醇激素受体结合的鉴别特征

Rashidian, Azam; Pitkänen, Sini; Maltarollo, Vinicius Goncalves; Schoppmeier, Ulrich; Shevchenko, Ekaterina; Medarametla, Prasanthi; Poso, Antti; Küblbeck, Jenni; Honkakoski, Paavo; Kronenberger, Thales

Thiazole Derivatives as Promising Candidates for Cryptococcosis Therapy

噻唑衍生物作为隐球菌病治疗的潜在候选药物

Leocádio, Victor Augusto Teixeira; Miranda, Isabela L; Magalhães, Martha H C; Dos Santos Júnior, Valtair Severino; Goncalves, José Eduardo; Oliveira, Renata Barbosa; Maltarollo, Vinicius Gonçalves; Bastos, Rafael Wesley; Goldman, Gustavo; Johann, Susana; Teixeira de Aguiar Peres, Nalu; Santos, Daniel de Assis

Can the interleukin TNF-α be used as a biomarker for pulp necrosis?

白细胞介素TNF-α能否用作牙髓坏死的生物标志物?

Brasil da Silva, Carlos Wesley Lopes; De Oliveira, Beatriz Melare; Duarte, Jheinis Stefany Pascuineli; Maltarollo, Thalya Fernanda Hortsh; Strazzi-Sahyon, Henrico Badaoui; Sivieri-Araújo, Gustavo

Understanding the Enzyme (S)-Norcoclaurine Synthase Promiscuity to Aldehydes and Ketones

了解 (S)-去甲劳林合酶对醛和酮的混杂性

Salvatti, Brunno A; Chagas, Marcelo A; Fernandes, Phillipe O; Ladeira, Yan F X; Bozzi, Aline S; Valadares, Veronica S; Valente, Ana Paula; de Miranda, Amanda S; Rocha, Willian R; Maltarollo, Vinicius G; Moraes, Adolfo H

A critical assessment of bioactive compounds databases

对生物活性化合物数据库的批判性评估

de Azevedo, Daniela Quadros; Campioni, Beatriz Mattos; Pedroz Lima, Felipe Augusto; L Medina-Franco, José; Castilho, Rachel Oliveira; Maltarollo, Vinícius Gonçalves

Trypanosoma cruzi Sirtuin 2 as a Relevant Druggable Target: New Inhibitors Developed by Computer-Aided Drug Design

克氏锥虫 Sirtuin 2 作为相关可用药靶点:通过计算机辅助药物设计开发的新型抑制剂

Glaucio Monteiro Ferreira, Thales Kronenberger, Vinicius Gonçalves Maltarollo, Antti Poso, Fernando de Moura Gatti, Vitor Medeiros Almeida, Sandro Roberto Marana, Carla Duque Lopes, Daiane Yukie Tezuka, Sérgio de Albuquerque, Flavio da Silva Emery, Gustavo Henrique Goulart Trossini