日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

CAMPER: mechanistic artificial intelligence for designing peptides that target MRSA persisters

CAMPER:用于设计靶向耐甲氧西林金黄色葡萄球菌(MRSA)持续感染肽的机制人工智能

Shehadeh, Fadi; Mishra, Biswajit; Ferrer-Espada, Raquel; Basu, Anindya; Felix, LewisOscar; Dellis, Charilaos; Ganesan, Narchonai; Zhang, Liyang; Martens, Andrew T; Goulev, Youlian; Sherman, Michael B; Paulsson, Johan; Naik, Mandar T; Sotiriadis, Paul P; Mylonakis, Eleftherios

Antimicrobial peptide developed with machine learning sequence optimization targets drug resistant Staphylococcus aureus in mice

利用机器学习序列优化技术开发的抗菌肽可靶向小鼠体内的耐药金黄色葡萄球菌。

Mishra, Biswajit; Basu, Anindya; Shehadeh, Fadi; Felix, LewisOscar; Kollala, Sai Sundeep; Chhonker, Yashpal Singh; Naik, Mandar T; Dellis, Charilaos; Zhang, Liyang; Ganesan, Narchonai; Murry, Daryl J; Gu, Jianhua; Sherman, Michael B; Ausubel, Frederick M; Sotiriadis, Paul P; Mylonakis, Eleftherios

The identification of a novel interaction site for the human immunodeficiency virus capsid on nucleoporin 153.

鉴定出人类免疫缺陷病毒衣壳与核孔蛋白 153 的新型相互作用位点

Li Shunji, Lund-Andersen Peik, Wang Szu-Huan, Ytreberg F Marty, Naik Mandar T, Patel Jagdish Suresh, Rowley Paul Andrew

Reciprocal antagonism of PIN1-APC/CCDH1 governs mitotic protein stability and cell cycle entry

PIN1-APC/CCDH1 的相互拮抗作用控制有丝分裂蛋白的稳定性和细胞周期进入

Shizhong Ke #, Fabin Dang #, Lin Wang #, Jia-Yun Chen #, Mandar T Naik, Wenxue Li, Abhishek Thavamani, Nami Kim, Nandita M Naik, Huaxiu Sui, Wei Tang, Chenxi Qiu, Kazuhiro Koikawa, Felipe Batalini, Emily Stern Gatof, Daniela Arango Isaza, Jaymin M Patel, Xiaodong Wang, John G Clohessy, Yujing J Heng

Syn3, a newly developed cyclic peptide and BDNF signaling enhancer, ameliorates retinal ganglion cell degeneration in diabetic retinopathy

Syn3 是一种新开发的环状肽和 BDNF 信号增强剂,可改善糖尿病视网膜病变中的视网膜神经节细胞变性。

Li, Ke-Ran; Huan, Meng-Jia; Yao, Jin; Li, Jia-Jun; Cao, Yuan; Wang, Suyu; Naik, Mandar T; Fang, Yuan; Marshall, John; Lan, Chang-Gong; Cao, Cong

Targeting the postsynaptic scaffolding protein PSD-95 enhances BDNF signaling to mitigate depression-like behaviors in mice

靶向突触后支架蛋白PSD-95可增强BDNF信号传导,从而减轻小鼠的抑郁样行为。

Shi, Xin; Zhou, Xiao-Zhong; Chen, Gang; Luo, Wei-Feng; Zhou, Chengyu; He, Tian-Ju; Naik, Mandar T; Jiang, Qin; Marshall, John; Cao, Cong

Structure-based design of peptidomimetic inhibitors of PSD-95 with improved affinity for the PDZ3 domain

基于结构的PSD-95肽模拟抑制剂设计,提高了其对PDZ3结构域的亲和力。

Naik, Mandar T; Naik, Nandita; Hu, Tony; Wang, Szu-Huan; Marshall, John

Activation of human RNA lariat debranching enzyme Dbr1 by binding protein TTDN1 occurs though an intrinsically disordered C-terminal domain

人类 RNA 套索脱支酶 Dbr1 被结合蛋白 TTDN1 激活,尽管 C 末端结构域本身无序

Nathaniel E Clark, Adam Katolik, Pascal Gallant, Anastasia Welch, Eileen Murphy, Luke Buerer, Christoph Schorl, Nandita Naik, Mandar T Naik, Stephen P Holloway, Kristin Cano, Susan T Weintraub, Katherine M Howard, P John Hart, Gerwald Jogl, Masad J Damha, William G Fairbrother

Structure-based development of new cyclic compounds targeting PSD-95 PDZ3 domain

基于结构的针对 PSD-95 PDZ3 结构域的新型环状化合物的开发

Mandar T Naik, Nandita Naik, Tony Hu, Szu-Huan Wang, John Marshall

Reciprocal inhibition of PIN1 and APC/CCDH1 controls timely G1/S transition and creates therapeutic vulnerability

PIN1 和 APC/CCDH1 的相互抑制可控制 G1/S 转换的及时性并造成治疗脆弱性

Shizhong Ke, Fabin Dang, Lin Wang, Jia-Yun Chen, Mandar T Naik, Abhishek Thavamani, Yansheng Liu, Wenxue Li, Nami Kim, Nandita M Naik, Huaxiu Sui, Wei Tang, Chenxi Qiu, Kazuhiro Koikawa, Felipe Batalini, Xiaodong Wang, John G Clohessy, Yujing Jan Heng, Galit Lahav, Nathanael S Gray, Xiao Zhen Zho, W