日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Antibacterial and Alkali-responsive Cationic Waterborne Polyurethane Based on Modification of Aloe Emodin

基于芦荟大黄素改性的抗菌碱性响应阳离子水性聚氨酯

Xiong, Xiaoyan; Li, Xiaobin; Zhu, Zifan; Zhang, Ending; Shi, Jun; Lu, Mangeng

Utilization of Metabolite Identification and Structural Data to Guide Design of Low-Dose IDO1 Inhibitors

利用代谢物鉴定和结构数据指导低剂量IDO1抑制剂的设计

Hopkins, Brett; Zhang, Hongjun; Bharathan, Indu; Li, Derun; Pu, Qinglin; Zhou, Hua; Martinot, Theodore A; Fradera, Xavier; Lammens, Alfred; Lesburg, Charles A; Cohen, Ryan D; Ballard, Jeanine; Knemeyer, Ian; Otte, Karin; Vincent, Stella; Miller, J Richard; Solban, Nicolas; Cheng, Mangeng; Geda, Prasanthi; Smotrov, Nadya; Song, Xuelei; Bennett, David Jonathan; Han, Yongxin

Carbamate and N-Pyrimidine Mitigate Amide Hydrolysis: Structure-Based Drug Design of Tetrahydroquinoline IDO1 Inhibitors

氨基甲酸酯和N-嘧啶可减轻酰胺水解:基于结构的四氢喹啉IDO1抑制剂药物设计

Li, Derun; Deng, Yongqi; Achab, Abdelghani; Bharathan, Indu; Hopkins, Brett Andrew; Yu, Wensheng; Zhang, Hongjun; Sanyal, Sulagna; Pu, Qinglin; Zhou, Hua; Liu, Kun; Lim, Jongwon; Fradera, Xavier; Lesburg, Charles A; Lammens, Alfred; Martinot, Theodore A; Cohen, Ryan D; Doty, Amy C; Ferguson, Heidi; Nickbarg, Elliott B; Cheng, Mangeng; Spacciapoli, Peter; Geda, Prasanthi; Song, Xuelei; Smotrov, Nadya; Abeywickrema, Pravien; Andrews, Christine; Chamberlin, Chad; Mabrouk, Omar; Curran, Patrick; Richards, Matthew; Saradjian, Peter; Miller, J Richard; Knemeyer, Ian; Otte, Karin M; Vincent, Stella; Sciammetta, Nunzio; Pasternak, Alexander; Bennett, David Jonathan; Han, Yongxin

Structure-Based Discovery of Proline-Derived Arginase Inhibitors with Improved Oral Bioavailability for Immuno-Oncology

基于结构的脯氨酸衍生精氨酸酶抑制剂的发现及其在免疫肿瘤学中提高的口服生物利用度

Lu, Min; Zhang, Hongjun; Li, Derun; Childers, Matthew; Pu, Qinglin; Palte, Rachel L; Gathiaka, Symon; Lyons, Thomas W; Palani, Anandan; Fan, Peter W; Spacciapoli, Peter; Miller, J Richard; Cho, Hyelim; Cheng, Mangeng; Chakravarthy, Kalyan; O'Neil, Jennifer; Eangoor, Padmanabhan; Beard, Adam; Kim, Hai-Young; Saurí, Josep; Gunaydin, Hakan; Sloman, David L; Siliphaivanh, Phieng; Cumming, Jared; Fischer, Christian

Cancer-Associated Fibroblasts Promote Immunosuppression by Inducing ROS-Generating Monocytic MDSCs in Lung Squamous Cell Carcinoma

癌症相关成纤维细胞通过诱导肺鳞状细胞癌中产生 ROS 的单核细胞 MDSC 来促进免疫抑制

Handan Xiang, Carlo P Ramil #, Josephine Hai #, Chunsheng Zhang, Huijun Wang, Amanda A Watkins, Roshi Afshar, Peter Georgiev, Marc A Sze, Xuelei S Song, Patrick J Curran, Mangeng Cheng, J Richard Miller, Dongyu Sun, Andrey Loboda, Yanlin Jia, Lily Y Moy, An Chi, Philip E Brandish

Strategic Incorporation of Polarity in Heme-Displacing Inhibitors of Indoleamine-2,3-dioxygenase-1 (IDO1)

策略性地将极性引入血红素置换抑制剂中,以抑制吲哚胺-2,3-双加氧酶-1 (IDO1)

White, Catherine; McGowan, Meredeth A; Zhou, Hua; Sciammetta, Nunzio; Fradera, Xavier; Lim, Jongwon; Joshi, Elizabeth M; Andrews, Christine; Nickbarg, Elliott B; Cowley, Phillip; Trewick, Sarah; Augustin, Martin; von Köenig, Konstanze; Lesburg, Charles A; Otte, Karin; Knemeyer, Ian; Woo, Hyun; Yu, Wensheng; Cheng, Mangeng; Spacciapoli, Peter; Geda, Prasanthi; Song, Xuelei; Smotrov, Nadya; Curran, Patrick; Heo, Mee Ra; Abeywickrema, Pravien; Miller, J Richard; Bennett, David Jonathan; Han, Yongxin

Discovery and Optimization of Rationally Designed Bicyclic Inhibitors of Human Arginase to Enhance Cancer Immunotherapy

发现和优化合理设计的双环人精氨酸酶抑制剂以增强癌症免疫疗法

Mitcheltree, Matthew J; Li, Derun; Achab, Abdelghani; Beard, Adam; Chakravarthy, Kalyan; Cheng, Mangeng; Cho, Hyelim; Eangoor, Padmanabhan; Fan, Peter; Gathiaka, Symon; Kim, Hai-Young; Lesburg, Charles A; Lyons, Thomas W; Martinot, Theodore A; Miller, J Richard; McMinn, Spencer; O'Neil, Jennifer; Palani, Anandan; Palte, Rachel L; Saurí, Josep; Sloman, David L; Zhang, Hongjun; Cumming, Jared N; Fischer, Christian

Discovery of Potent and Orally Available Bicyclo[1.1.1]pentane-Derived Indoleamine-2,3-dioxygenase 1 (IDO1) Inhibitors

发现高效且口服有效的双环[1.1.1]戊烷衍生的吲哚胺-2,3-双加氧酶1 (IDO1) 抑制剂

Pu, Qinglin; Zhang, Hongjun; Guo, Liangqin; Cheng, Mangeng; Doty, Amy C; Ferguson, Heidi; Fradera, Xavier; Lesburg, Charles A; McGowan, Meredeth A; Miller, J Richard; Geda, Prasanthi; Song, Xuelei; Otte, Karin; Sciammetta, Nunzio; Solban, Nicolas; Yu, Wensheng; Sloman, David L; Zhou, Hua; Lammens, Alfred; Neumann, Lars; Bennett, David Jonathan; Pasternak, Alexander; Han, Yongxin

Discovery of Amino-cyclobutarene-derived Indoleamine-2,3-dioxygenase 1 (IDO1) Inhibitors for Cancer Immunotherapy

发现氨基环丁烯衍生的吲哚胺-2,3-双加氧酶1 (IDO1) 抑制剂用于癌症免疫治疗

Zhang, Hongjun; Liu, Kun; Pu, Qinglin; Achab, Abdelghani; Ardolino, Michael J; Cheng, Mangeng; Deng, Yongqi; Doty, Amy C; Ferguson, Heidi; Fradera, Xavier; Knemeyer, Ian; Kurukulasuriya, Ravi; Lam, Yu-Hong; Lesburg, Charles A; Martinot, Theodore A; McGowan, Meredeth A; Miller, J Richard; Otte, Karin; Biju, Purakattle J; Sciammetta, Nunzio; Solban, Nicolas; Yu, Wensheng; Zhou, Hua; Wang, Xiao; Bennett, David Jonathan; Han, Yongxin

Therapeutic efficacy of the bromodomain inhibitor OTX015/MK-8628 in ALK-positive anaplastic large cell lymphoma: an alternative modality to overcome resistant phenotypes

溴结构域抑制剂 OTX015/MK-8628 对 ALK 阳性间变性大细胞淋巴瘤的治疗效果:克服耐药表型的替代方法

Michela Boi, Maria Todaro, Valentina Vurchio, Shao Ning Yang, John Moon, Ivo Kwee, Andrea Rinaldi, Heng Pan, Ramona Crescenzo, Mangeng Cheng, Leandro Cerchietti, Olivier Elemento, Maria E Riveiro, Esteban Cvitkovic, Francesco Bertoni, Giorgio Inghirami; AIRC 5xMille Consortium ‘Genetics-Driven Targe