日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Efficacy of HMJ-38, a new quinazolinone analogue, against the gemcitabine-resistant MIA-PaCa-2 pancreatic cancer cells

新型喹唑啉酮类似物 HMJ-38 对吉西他滨耐药 MIA-PaCa-2 胰腺癌细胞的疗效

Mann-Jen Hour, Fuu-Jen Tsai, I-Lu Lai, Je-Wei Tsao, Jo-Hua Chiang, Yu-Jen Chiu, Hsing-Fang Lu, Yu-Ning Juan, Jai-Sing Yang, Shih-Chang Tsai1

Glycyrrhizic Acid Derivatives Bearing Amino Acid Residues in the Carbohydrate Part as Dengue Virus E Protein Inhibitors: Synthesis and Antiviral Activity

糖基部分含氨基酸残基的甘草酸衍生物作为登革病毒E蛋白抑制剂的合成及抗病毒活性

Mann-Jen Hour, Yeh Chen, Chen-Sheng Lin, Lidia A Baltina, Ju-Ying Kan, Yan-Ting Tsai, Yan-Tung Kiu, Hsueh-Chou Lai, Lia A Baltina, Svetlana F Petrova, Cheng-Wen Lin

Novel quinazolinone MJ‑33 induces AKT/mTOR‑mediated autophagy‑associated apoptosis in 5FU‑resistant colorectal cancer cells

新型喹唑啉酮 MJ-33 诱导 5FU 耐药结直肠癌细胞中 AKT/mTOR 介导的自噬相关细胞凋亡

Hai-Anh Ha, Jo-Hua Chiang, Fuu-Jen Tsai, Da-Tian Bau, Yu-Ning Juan, Yu-Hsiang Lo, Mann-Jen Hour, Jai-Sing Yang

Disruption of IGF‑1R signaling by a novel quinazoline derivative, HMJ‑30, inhibits invasiveness and reverses epithelial-mesenchymal transition in osteosarcoma U‑2 OS cells

新型喹唑啉衍生物 HMJ-30 阻断 IGF-1R 信号传导,可抑制骨肉瘤 U-2 OS 细胞的侵袭性并逆转上皮-间质转化

Yu-Jen Chiu, Mann-Jen Hour, Yi-An Jin, Chi-Cheng Lu, Fuu-Jen Tsai, Tai-Lin Chen, Hsu Ma, Yu-Ning Juan, Jai-Sing Yang

Single-Round Infectious Particle Antiviral Screening Assays for the Japanese Encephalitis Virus

日本脑炎病毒单轮感染性颗粒抗病毒筛选试验

Chien-Yi Lu, Mann-Jen Hour, Ching-Ying Wang, Su-Hua Huang, Wen-Xiang Mu, Yu-Chun Chang, Cheng-Wen Lin

Tubacin, an HDAC6 Selective Inhibitor, Reduces the Replication of the Japanese Encephalitis Virus via the Decrease of Viral RNA Synthesis

Tubacin 是一种 HDAC6 选择性抑制剂,它通过减少病毒 RNA 合成来减少日本脑炎病毒的复制

Chien-Yi Lu, Yi-Chih Chang, Chun-Hung Hua, Chieh Chuang, Su-Hua Huang, Szu-Hao Kung, Mann-Jen Hour, Cheng-Wen Lin

MJ-66 induces malignant glioma cells G2/M phase arrest and mitotic catastrophe through regulation of cyclin B1/Cdk1 complex

MJ-66 通过调节细胞周期蛋白 B1/Cdk1 复合物诱导恶性胶质瘤细胞 G2/M 期停滞和有丝分裂灾难

Wei-Ting Liu, Ching Chen, I-Chen Lu, Sheng-Chu Kuo, Kuo-Hsiung Lee, Tai-Lin Chen, Ta-Shu Song, Yi-Liang Lu, Po-Wu Gean, Mann-Jen Hour

5-Lipoxygenase inhibitors attenuate TNF-α-induced inflammation in human synovial fibroblasts

5-脂氧合酶抑制剂可减轻人类滑膜成纤维细胞中 TNF-α 诱发的炎症

Han-Ching Lin, Tzu-Hung Lin, Ming-Yueh Wu, Yung-Cheng Chiu, Chih-Hsin Tang, Mann-Jen Hour, Houng-Chi Liou, Huang-Ju Tu, Rong-Sen Yang, Wen-Mei Fu