Identification of Structurally Novel KRAS(G12C) Inhibitors through Covalent DNA-Encoded Library Screening
通过共价DNA编码文库筛选鉴定结构新颖的KRAS(G12C)抑制剂
期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/acs.jmedchem.4c03071
Huang, David; Manoni, Francesco; Sun, Zhen; Liu, Rongfeng; Allen, Jennifer R; Banerjee, Abhisek; Cee, Victor J; Eshon, Josephine; Frohn, Michael J; Kaller, Matthew R; Lee, Heejun; Li, Cui; Li, Xun; Lopez, Patricia; Ma, Vu; Medina, Jose M; Mohr, Christopher; Mukhina, Olga A; Pickrell, Alexander J; Stellwagen, John; Wu, Wenting; Zhang, Wenhan; Zhu, Kai; Dahal, Upendra P; Hu, Liaoyuan A; Leavitt, Monica; Li, Wencui; Li, Yu; Ma, Yingli; Rex, Karen; Saiki, Anne Y; Wang, Paul; Sun, Yaping; Dai, Dongcheng; Tamayo, Nuria A; Lanman, Brian A