日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Effects of CT-388, a once-weekly signaling-biased dual GLP-1/GIP receptor agonist, on weight loss and glycemic control in preclinical models and participants with obesity

CT-388 是一种每周一次给药的信号传导偏向型双重 GLP-1/GIP 受体激动剂,本研究探讨了其对临床前模型和肥胖患者体重减轻和血糖控制的影响。

Chakravarthy, Manu V; Rodriguez, Ruben; Hergarden, Anne; Elliott, Michael A; Frias, Juan P; Argüelles-Tello, Federico A; Tenorio, Edgar; Rankin, Jonathan E; Wu, Jingtao; Krishnan, Shyam; Erlanson, Daniel A; Fucini, Raymond V; Bone, Derek; Iwig, Jeffrey S; Acosta, Luis; Untereiner, Ashley; Pant, Asmita; Patton, Avalon; Sanchez-Sanchez, Leyla L; Luo, Jian; Steinberg, Alexandra; Bialonczyk, Damian; Hansen, Stig K

Efficacy and safety of CT-868, a novel, fully biased, dual glucagon-like peptide-1/glucose-dependent insulinotropic polypeptide receptor agonist, in type 2 diabetes: A double-blind, randomized placebo controlled phase 2 trial

CT-868(一种新型的、完全偏向性的双重胰高血糖素样肽-1/葡萄糖依赖性促胰岛素多肽受体激动剂)治疗2型糖尿病的疗效和安全性:一项双盲、随机、安慰剂对照的II期试验

Chakravarthy, Manu V; Elliott, Michael A; Acosta, Luis; Sonnenberg, Gabriele E; Bialonczyk, Damian; Wu, Jingtao; Argüelles-Tello, Federico A; Garcia-Reza, Raymundo; González-González, José Gerardo; Hansen, Stig K; Frias, Juan P

Bill Scott (1963–2025)

比尔·斯科特(1963–2025)

Manu, V S; Melacini, Giuseppe; Kovrigin, Evgenii L; Loria, J Patrick; Veglia, Gianluigi; Noller, Harry F

Biased agonism of GLP-1R and GIPR enhances glucose lowering and weight loss, with dual GLP-1R/GIPR biased agonism yielding greater efficacy.

GLP-1R 和 GIPR 的偏向性激动作用可增强降血糖和减肥效果,而 GLP-1R/GIPR 的双重偏向性激动作用可产生更大的疗效

Rodriguez Ruben, Hergarden Anne, Krishnan Shyam, Morales Marikris, Lam Davina, Tracy Ted, Tang Teresa, Patton Avalon, Lee Craig, Pant Asmita, Erlanson Daniel A, Enquist Johan, Bone Derek, Fucini Ray, Bialonczyk Damian, Hansen Stig K, Luo Jian, Chakravarthy Manu V

Protein Kinase A Phosphorylates a Conformationally High-energy State of Raf Kinase Inhibitory Protein

蛋白激酶A磷酸化Raf激酶抑制蛋白的构象高能状态。

Olivieri, Cristina; Biancaniello, Carmen; Manu, V S; Walters, Matthew Steven; Masterson, Larry; Rosner, Marsha Rich; De Simone, Alfonso; Veglia, Gianluigi

Prevalence and Predictors of Follow-up Endoscopic Biopsy in Patients With Celiac Disease in the United States

美国乳糜泻患者随访内镜活检的患病率及预测因素

Venkat, Manu V; Chen, Ling; Wright, Jason D; Lebwohl, Benjamin

Assessment of Serum Ferritin Levels in Female Patients With Telogen Effluvium

对患有休止期脱发的女性患者血清铁蛋白水平的评估

Thamotharan, Nishantan; Harikumar, Manu V; Sundaram, Murugan; Swaminathan, Adikrishnan; Rangarajan, Sudha

AI-designed NMR spectroscopy RF pulses for fast acquisition at high and ultra-high magnetic fields

人工智能设计的核磁共振波谱射频脉冲,可在高磁场和超高磁场下实现快速采集

Manu, V S; Olivieri, Cristina; Veglia, Gianluigi

Water irradiation devoid pulses enhance the sensitivity of (1)H,(1)H nuclear Overhauser effects

无脉冲水辐照可增强 (1)H,(1)H 核奥弗豪瑟效应的灵敏度

Manu, V S; Olivieri, Cristina; Veglia, Gianluigi

Reconfigurable halide perovskite nanocrystal memristors for neuromorphic computing

用于神经形态计算的可重构卤化物钙钛矿纳米晶忆阻器

John, Rohit Abraham; Demirağ, Yiğit; Shynkarenko, Yevhen; Berezovska, Yuliia; Ohannessian, Natacha; Payvand, Melika; Zeng, Peng; Bodnarchuk, Maryna I; Krumeich, Frank; Kara, Gökhan; Shorubalko, Ivan; Nair, Manu V; Cooke, Graham A; Lippert, Thomas; Indiveri, Giacomo; Kovalenko, Maksym V