Truncated (N)-Methanocarba Nucleosides as Partial Agonists at Mouse and Human A3 Adenosine Receptors: Affinity Enhancement by N6-(2-Phenylethyl) Substitution
截短的 (N)-亚甲基羰基核苷作为小鼠和人类 A3 腺苷受体的部分激动剂:通过 N6-(2-苯乙基) 取代增强亲和力
期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/acs.jmedchem.0c00235
Dilip K Tosh, Veronica Salmaso, Harsha Rao, Amelia Bitant, Courtney L Fisher, David I Lieberman, Helmut Vorbrüggen, Marc L Reitman, Oksana Gavrilova, Zhan-Guo Gao, John A Auchampach, Kenneth A Jacobson