日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Covalent Modification of p53 by (E)-1-(4-Methylpiperazin-1-yl)-3-(5-nitrofuran-2-yl)prop-2-en-1-one

(E)-1-(4-甲基哌嗪-1-基)-3-(5-硝基呋喃-2-基)丙-2-烯-1-酮对p53的共价修饰

Kate Brown,Marco Robello,Andrew J Perciaccante,Jerry C Dinan,Tapan K Maity,Gaelyn C Lyons,Jay P Kumar,Stewart R Durell,Harichandra D Tagad,Daniel Schilling,Herman Nikolayevskiy,Robert O'Connor,Ettore Appella,Daniel H Appella,Lisa M Jenkins

Alkyl-substituted N-methylaryl-N'-aryl-4-aminobenzamides: A new series of small molecule inhibitors for Wip1 phosphatase

烷基取代的 N-甲基芳基-N'-芳基-4-氨基苯甲酰胺:一系列新型 Wip1 磷酸酶小分子抑制剂

Marco Robello, Hongchao Zheng, Mrinmoy Saha, Kara M George Rosenker, Subrata Debnath, Jay Prakash Kumar, Harichandra D Tagad, Sharlyn J Mazur, Ettore Appella, Daniel H Appella

The structure-activity profile of mercaptobenzamides' anti-HIV activity suggests that thermodynamics of metabolism is more important than binding affinity to the target

巯基苯甲酰胺抗 HIV 活性的结构-活性特征表明,代谢热力学比与靶标的结合亲和力更重要

Herman Nikolayevskiy, Marco Robello, Michael T Scerba, Evan H Pasternak, Mrinmoy Saha, Tracy L Hartman, Caitlin A Buchholz, Robert W Buckheit Jr, Stewart R Durell, Daniel H Appella