日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Activation of CAMK2 by pseudokinase PEAK1 represents a targetable pathway in triple negative breast cancer

假激酶 PEAK1 激活 CAMK2 是三阴性乳腺癌中可靶向的通路

Xue Yang, Xiuquan Ma, Tianyue Zhao, David R Croucher, Elizabeth V Nguyen, Kimberley C Clark, Changyuan Hu, Sharissa L Latham, Charles Bayly-Jones, Bao V Nguyen, Srikanth Budnar, Sung-Young Shin, Lan K Nguyen, Thomas R Cotton, Anderly C Chüeh, Terry C C Lim Kam Sian, Margaret M Stratton, Andrew M Ell

Ligand-induced CaMKIIα hub Trp403 flip, hub domain stacking, and modulation of kinase activity

配体诱导的 CaMKIIα 枢纽 Trp403 翻转、枢纽域堆积和激酶活性调节

Dilip Narayanan, Anne Sofie G Larsen, Stine Juul Gauger, Ruth Adafia, Rikke Bartschick Hammershøi, Louise Hamborg, Jesper Bruus-Jensen, Nane Griem-Krey, Christine L Gee, Bente Frølund, Margaret M Stratton, John Kuriyan, Jette Sandholm Kastrup, Annette E Langkilde, Petrine Wellendorph, Sara M Ø Solba

Reciprocal Activation within a Kinase-Effector Complex Underlying Persistence of Structural LTP

激酶效应复合物内的相互激活是结构性 LTP 持久性的基础

Takeo Saneyoshi, Hitomi Matsuno, Akio Suzuki, Hideji Murakoshi, Nathan G Hedrick, Emily Agnello, Rory O'Connell, Margaret M Stratton, Ryohei Yasuda, Yasunori Hayashi

Molecular mechanism of activation-triggered subunit exchange in Ca(2+)/calmodulin-dependent protein kinase II

钙/钙调蛋白依赖性蛋白激酶Ⅱ活化引发亚基交换的分子机制

Moitrayee Bhattacharyya, Margaret M Stratton, Catherine C Going, Ethan D McSpadden, Yongjian Huang, Anna C Susa, Anna Elleman, Yumeng Melody Cao, Nishant Pappireddi, Pawel Burkhardt, Christine L Gee, Tiago Barros, Howard Schulman, Evan R Williams, John Kuriyan

A mechanism for tunable autoinhibition in the structure of a human Ca2+/calmodulin- dependent kinase II holoenzyme

人类 Ca2+/钙调蛋白依赖性激酶 II 全酶结构中可调节的自抑制机制

Luke H Chao, Margaret M Stratton, Il-Hyung Lee, Oren S Rosenberg, Joshua Levitz, Daniel J Mandell, Tanja Kortemme, Jay T Groves, Howard Schulman, John Kuriyan