Synthesis and biological evaluation of 2-amino-3-(3',4',5'-trimethoxybenzoyl)-6-substituted-4,5,6,7-tetrahydrothieno[2,3-c]pyridine derivatives as antimitotic agents and inhibitors of tubulin polymerization
2-氨基-3-(3',4',5'-三甲氧基苯甲酰基)-6-取代-4,5,6,7-四氢噻吩并[2,3-c]吡啶衍生物的合成及生物学评价,作为抗有丝分裂剂和微管蛋白聚合抑制剂
期刊:Bioorganic & Medicinal Chemistry Letters
影响因子:2.2
doi:10.1016/j.bmcl.2008.08.006
Romagnoli, Romeo; Baraldi, Pier Giovanni; Carrion, Maria Dora; Cruz-Lopez, Olga; Cara, Carlota Lopez; Tolomeo, Manlio; Grimaudo, Stefania; Di Cristina, Antonietta; Pipitone, Maria Rosa; Balzarini, Jan; Kandil, Sahar; Brancale, Andrea; Sarkar, Taradas; Hamel, Ernest