Discovery of highly selective and orally active lysophosphatidic acid receptor-1 antagonists with potent activity on human lung fibroblasts
发现具有高选择性和口服活性的溶血磷脂酸受体-1拮抗剂,对人肺成纤维细胞具有强效活性
期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/jm301022v
Yimin Qian, Matthew Hamilton, Achyutharao Sidduri, Stephen Gabriel, Yonglin Ren, Ruoqi Peng, Rama Kondru, Arjun Narayanan, Terry Truitt, Rachid Hamid, Yun Chen, Lin Zhang, Adrian J Fretland, Ruben Alvarez Sanchez, Kung-Ching Chang, Matthew Lucas, Ryan C Schoenfeld, Dramane Laine, Maria E Fuentes, Ch