日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Targeting Viral and Cellular Cysteine Proteases for Treatment of New Variants of SARS-CoV-2

针对病毒和细胞半胱氨酸蛋白酶治疗 SARS-CoV-2 新变种

Davide Gentile, Lucia Chiummiento, Alessandro Santarsiere, Maria Funicello, Paolo Lupattelli, Antonio Rescifina, Assunta Venuti, Anna Piperno, Maria Teresa Sciortino, Rosamaria Pennisi

PEGylated Liposomes Loaded with Carbamate Inhibitor ANP0903 Trigger Apoptosis by Enhancing ER Stress in HepG2 Cancer Cells

载有氨基甲酸酯抑制剂 ANP0903 的聚乙二醇化脂质体通过增强 HepG2 癌细胞中的 ER 应激来引发细胞凋亡

Carla Caddeo, Rocchina Miglionico, Roberta Rinaldi, Ilaria Nigro, Daniela Lamorte, Lucia Chiummiento, Paolo Lupattelli, Maria Funicello, Rosarita D'Orsi, Donatella Valenti, Valentina Santoro, Anna Maria Fadda, Faustino Bisaccia, Antonio Vassallo, Maria Francesca Armentano

Two Novel Precursors of the HIV-1 Protease Inhibitor Darunavir Target the UPR/Proteasome System in Human Hepatocellular Carcinoma Cell Line HepG2

HIV-1 蛋白酶抑制剂达芦那韦的两种新型前体靶向人类肝癌细胞系 HepG2 中的 UPR/蛋白酶体系统

Roberta Rinaldi, Rocchina Miglionico, Ilaria Nigro, Rosarita D'Orsi, Lucia Chiummiento, Maria Funicello, Paolo Lupattelli, Ilaria Laurenzana, Alessandro Sgambato, Magnus Monné, Faustino Bisaccia, Maria Francesca Armentano

The Pseudo-Symmetric N-benzyl Hydroxyethylamine Core in a New Series of Heteroarylcarboxyamide HIV-1 Pr Inhibitors: Synthesis, Molecular Modeling and Biological Evaluation

新型杂芳基羧酰胺 HIV-1 Pr 抑制剂系列中的伪对称 N-苄基羟乙胺核心:合成、分子建模和生物学评价

Rosarita D'Orsi, Maria Funicello, Teresa Laurita, Paolo Lupattelli, Federico Berti, Lucia Chiummiento

One Pot Synthesis of Micromolar BACE-1 Inhibitors Based on the Dihydropyrimidinone Scaffold and Their Thia and Imino Analogues

基于二氢嘧啶酮骨架及其硫杂和亚氨基类似物的微摩尔 BACE-1 抑制剂的一锅合成

Jessica Bais, Fabio Benedetti, Federico Berti, Iole Cerminara, Sara Drioli, Maria Funicello, Giorgia Regini, Mattia Vidali, Fulvia Felluga

New synthesized polyoxygenated diarylheptanoids suppress lipopolysaccharide-induced neuroinflammation

新合成的多氧二芳基庚烷可抑制脂多糖诱导的神经炎症

Anna Santarsiero, Antonella Bochicchio, Maria Funicello, Paolo Lupattelli, Sabine Choppin, Françoise Colobert, Gilles Hanquet, Lucie Schiavo, Paolo Convertini, Lucia Chiummiento, Vittoria Infantino