日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

G protein-specific mechanisms in the serotonin 5-HT2A receptor regulate psychosis-related effects and memory deficits

血清素 5-HT2A 受体中的 G 蛋白特异性机制调节精神病相关影响和记忆缺陷

Elk Kossatz #, Rebeca Diez-Alarcia #, Supriya A Gaitonde, Carla Ramon-Duaso, Tomasz Maciej Stepniewski, David Aranda-Garcia, Itziar Muneta-Arrate, Elodie Tepaz, Suwipa Saen-Oon, Robert Soliva, Aida Shahraki, David Moreira, Jose Brea, Maria Isabel Loza, Rafael de la Torre, Peter Kolb, Michel Bouvier,

Fluorescence based HTS-compatible ligand binding assays for dopamine D3 receptors in baculovirus preparations and live cells

基于荧光的 HTS 兼容配体结合试验,用于检测杆状病毒制剂和活细胞中的多巴胺 D3 受体

Maris-Johanna Tahk, Tõnis Laasfeld, Elo Meriste, Jose Brea, Maria Isabel Loza, Maria Majellaro, Marialessandra Contino, Eddy Sotelo, Ago Rinken

From Serendipity to Rational Identification of the 5,6,7,8-Tetrahydrobenzo[4,5]thieno[2,3- d]pyrimidin-4(3 H)-one Core as a New Chemotype of AKT1 Inhibitors for Acute Myeloid Leukemia

从偶然发现到合理鉴定 5,6,7,8-四氢苯并[4,5]噻吩并[2,3- d]嘧啶-4(3 H)-酮核心为治疗急性髓系白血病的 AKT1 抑制剂新化学型

Andrea Astolfi, Francesca Milano, Deborah Palazzotti, Jose Brea, Maria Chiara Pismataro, Mariangela Morlando, Oriana Tabarrini, Maria Isabel Loza, Serena Massari, Maria Paola Martelli, Maria Letizia Barreca

Docking Screens for Dual Inhibitors of Disparate Drug Targets for Parkinson's Disease

帕金森病不同药物靶点的双重抑制剂对接筛选

Mariama Jaiteh, Alexey Zeifman, Marcus Saarinen, Per Svenningsson, Jose Bréa, Maria Isabel Loza, Jens Carlsson