9H-purine scaffold reveals induced-fit pocket plasticity of the BRD9 bromodomain
9H-嘌呤支架揭示了 BRD9 溴结构域的诱导契合口袋可塑性
期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/jm501893k
Sarah Picaud, Maria Strocchia, Stefania Terracciano, Gianluigi Lauro, Jacqui Mendez, Danette L Daniels, Raffaele Riccio, Giuseppe Bifulco, Ines Bruno, Panagis Filippakopoulos