日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Fixed combination of palmitoylethanolamide and melatonin in preventive therapy of migraine: results from a randomized clinical trial

棕榈酰乙醇胺和褪黑素固定组合用于偏头痛预防治疗:一项随机临床试验的结果

Piccolo, Vincenzo; Marzocchi, Adua; Maisto, Maria; Summa, Vincenzo; Tenore, Gian Carlo; Amoresano, Angela

Discovery of CDC42 Inhibitors with a Favorable Pharmacokinetic Profile and Anticancer In Vivo Efficacy

发现具有良好药代动力学特征和抗癌体内功效的 CDC42 抑制剂

Nicoletta Brindani, Linh M Vuong, Maria Antonietta La Serra, Noel Salvador, Andrea Menichetti, Isabella Maria Acquistapace, Jose Antonio Ortega, Marina Veronesi, Sine Mandrup Bertozzi, Maria Summa, Stefania Girotto, Rosalia Bertorelli, Andrea Armirotti, Anand K Ganesan, Marco De Vivo

Design, Synthesis, In Vitro and In Vivo Characterization of CDC42 GTPase Interaction Inhibitors for the Treatment of Cancer

用于治疗癌症的 CDC42 GTPase 相互作用抑制剂的设计、合成、体外和体内表征

Nicoletta Brindani, Linh M Vuong, Isabella Maria Acquistapace, Maria Antonietta La Serra, José Antonio Ortega, Marina Veronesi, Sine Mandrup Bertozzi, Maria Summa, Stefania Girotto, Rosalia Bertorelli, Andrea Armirotti, Anand K Ganesan, Marco De Vivo

Plant-Based, Hydrogel-like Microfibers as an Antioxidant Platform for Skin Burn Healing

植物基水凝胶状微纤维作为皮肤烧伤愈合的抗氧化平台

Fabrizio Fiorentini, Giulia Suarato, Maria Summa, Dalila Miele, Giuseppina Sandri, Rosalia Bertorelli, Athanassia Athanassiou

Structure-based design of CDC42 effector interaction inhibitors for the treatment of cancer

基于结构的设计用于治疗癌症的 CDC42 效应相互作用抑制剂

Sohail Jahid, Jose A Ortega, Linh M Vuong, Isabella Maria Acquistapace, Stephanie J Hachey, Jessica L Flesher, Maria Antonietta La Serra, Nicoletta Brindani, Giuseppina La Sala, Jacopo Manigrasso, Jose M Arencibia, Sine Mandrup Bertozzi, Maria Summa, Rosalia Bertorelli, Andrea Armirotti, Rongsheng J

Innovative Non-PrP-Targeted Drug Strategy Designed to Enhance Prion Clearance

旨在增强朊病毒清除能力的创新非PrP靶向药物策略

Arianna Colini Baldeschi, Marco Zattoni, Silvia Vanni, Lea Nikolic, Chiara Ferracin, Giuseppina La Sala, Maria Summa, Rosalia Bertorelli, Sine Mandrup Bertozzi, Gabriele Giachin, Paolo Carloni, Maria Laura Bolognesi, Marco De Vivo, Giuseppe Legname

Design, Synthesis, Dynamic Docking, Biochemical Characterization, and in Vivo Pharmacokinetics Studies of Novel Topoisomerase II Poisons with Promising Antiproliferative Activity

具有良好抗增殖活性的新型拓扑异构酶 II 毒物的设计、合成、动态对接、生化表征及体内药代动力学研究

Jose M Arencibia, Nicoletta Brindani, Sebastian Franco-Ulloa, Michela Nigro, Jissy Akkarapattiakal Kuriappan, Giuliana Ottonello, Sine Mandrup Bertozzi, Maria Summa, Stefania Girotto, Rosalia Bertorelli, Andrea Armirotti, Marco De Vivo

Novel, Potent, and Druglike Tetrahydroquinazoline Inhibitor That Is Highly Selective for Human Topoisomerase II α over β

新型、有效且类似药物的四氢喹唑啉抑制剂,对人类拓扑异构酶 II α 比 β 具有更高的选择性

Jose Antonio Ortega, Jose M Arencibia, Elirosa Minniti, Jo Ann W Byl, Sebastian Franco-Ulloa, Marco Borgogno, Vito Genna, Maria Summa, Sine Mandrup Bertozzi, Rosalia Bertorelli, Andrea Armirotti, Anna Minarini, Claudia Sissi, Neil Osheroff, Marco De Vivo

Design, Synthesis, and Biological Evaluation of a Series of Oxazolone Carboxamides as a Novel Class of Acid Ceramidase Inhibitors

一系列恶唑酮酰胺作为新型酸性神经酰胺酶抑制剂的设计、合成及生物学评价

Samantha Caputo, Simona Di Martino, Vincenzo Cilibrasi, Piero Tardia, Marco Mazzonna, Debora Russo, Ilaria Penna, Maria Summa, Sine Mandrup Bertozzi, Natalia Realini, Natasha Margaroli, Marco Migliore, Giuliana Ottonello, Min Liu, Peter Lansbury, Andrea Armirotti, Rosalia Bertorelli, Soumya S Ray, R

Improved Selective Class I HDAC and Novel Selective HDAC3 Inhibitors: Beyond Hydroxamic Acids and Benzamides

改良型选择性I类HDAC抑制剂和新型选择性HDAC3抑制剂:超越羟肟酸和苯甲酰胺

Bresciani, Alberto; Ontoria, Jesus M; Biancofiore, Ilaria; Cellucci, Antonella; Ciammaichella, Alina; Di Marco, Annalise; Ferrigno, Federica; Francone, Alessandra; Malancona, Savina; Monteagudo, Edith; Nizi, Emanuela; Pace, Paola; Ponzi, Simona; Rossetti, Ilaria; Veneziano, Maria; Summa, Vincenzo; Harper, Steven