日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Dysregulation of human ClpP using small molecules with piperazine-based scaffold for diffuse intrinsic pontine glioma therapy validated by patient-derived tumor organoids

利用哌嗪骨架小分子调控人ClpP失调治疗弥漫性内生性脑桥胶质瘤,并通过患者来源的肿瘤类器官验证其疗效

Miciaccia, Morena; Armenise, Domenico; Baldelli, Olga Maria; Liturri, Anselma; Mammone, Mariachiara; Graziano, Giovanni; Contino, Marialessandra; Rizzo, Francesca; Polosa, Paola Loguercio; Bruni, Francesco; Deligne, Clémence; Broutier, Laura; Cavallaro, Gianfranco; Fortuna, Cosimo Gianluca; Tolomeo, Anna; Green, Cadell; Bonifazi, Alessandro; Majaesic, Emily; Barghash, Marim M; Lee, Nok Pang Josh; Houry, Walid A; Gratteri, Carmen; Talarico, Carmine; Filieri, Silvana; Micalizzi, Giuseppe; Donnarumma, Danilo; Dugo, Paola; Mondello, Luigi; Sardanelli, Anna Maria; Nazarian, Javad; Ferorelli, Savina; Perrone, Maria Grazia; Scilimati, Antonio

Interactions of proteins with heparan sulfate

蛋白质与硫酸乙酰肝素的相互作用

Alotaibi, Faizah S; Alsadun, Marim M R; Alsaiari, Sarah A; Ramakrishnan, Krithika; Yates, Edwin A; Fernig, David G

Potent ClpP agonists with anticancer properties bind with improved structural complementarity and alter the mitochondrial N-terminome

具有抗癌特性的强效 ClpP 激动剂与改进的结构互补性结合并改变线粒体的 N 端

Mark F Mabanglo, Keith S Wong, Marim M Barghash, Elisa Leung, Stephanie H W Chuang, Afshan Ardalan, Emily M Majaesic, Cassandra J Wong, Shen Zhang, Henk Lang, Donald S Karanewsky, Andrew A Iwanowicz, Lee M Graves, Edwin J Iwanowicz, Anne-Claude Gingras, Walid A Houry

Cellular functions of the ClpP protease impacting bacterial virulence

ClpP蛋白酶的细胞功能影响细菌毒力

Aljghami, Mazen E; Barghash, Marim M; Majaesic, Emily; Bhandari, Vaibhav; Houry, Walid A

Aβ43 aggregates exhibit enhanced prion-like seeding activity in mice

Aβ43聚集体在小鼠体内表现出增强的朊病毒样播种活性。

Alejandro Ruiz-Riquelme ,Alison Mao ,Marim M Barghash ,Heather H C Lau ,Erica Stuart ,Gabor G Kovacs ,K Peter R Nilsson ,Paul E Fraser ,Gerold Schmitt-Ulms ,Joel C Watts

Development of Antibiotics That Dysregulate the Neisserial ClpP Protease

开发能扰乱奈瑟菌ClpP蛋白酶活性的抗生素

Binepal, Gursonika; Mabanglo, Mark F; Goodreid, Jordan D; Leung, Elisa; Barghash, Marim M; Wong, Keith S; Lin, Funing; Cossette, Michele; Bansagi, Jazmin; Song, Boxi; Balasco Serrão, Vitor Hugo; Pai, Emil F; Batey, Robert A; Gray-Owen, Scott D; Houry, Walid A

ClpP protease activation results from the reorganization of the electrostatic interaction networks at the entrance pores.

ClpP 蛋白酶的激活是由于入口孔处静电相互作用网络的重组所致

Mabanglo Mark F, Leung Elisa, Vahidi Siavash, Seraphim Thiago V, Eger Bryan T, Bryson Steve, Bhandari Vaibhav, Zhou Jin Lin, Mao Yu-Qian, Rizzolo Kamran, Barghash Marim M, Goodreid Jordan D, Phanse Sadhna, Babu Mohan, Barbosa Leandro R S, Ramos Carlos H I, Batey Robert A, Kay Lewis E, Pai Emil F, Houry Walid A