日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

A Chemical-Genetic Interaction Matrix Reveals Drug Mechanism and Genetic Architecture

化学-遗传相互作用矩阵揭示药物机制和遗传结构

Coulombe-Huntington, Jasmin; Bertomeu, Thierry; Huard, Caroline; Chatr-Aryamontri, Andrew; St-Cyr, Daniel J; Sánchez-Osuna, María; Papadopoli, David; Normandin, Karine; Paydar, Mohammadjavad; McLaughlan, Shannon; St-Denis, Corinne; Zhang, Li; Say, Henry; Palou, Roger; Stark, Chris; Breitkreutz, Bobby-Joe; van der Sloot, Almer M; Manohar, Sandhya; Lavoie, Hugo; Borden, Katherine L B; Raught, Brian; D'Amours, Damien; Sicheri, Frank; Verreault, Alain; Mader, Sylvie; Meloche, Sylvain; Therrien, Marc; Thibault, Pierre; Wilhelm, Brian; Dirks, Peter B; Aitchison, John D; Patton, Elizabeth; King, Randall W; Roux, Philippe P; Sauvageau, Guy; Hoang, Trang; Marinier, Anne; Harrington, Lea; Kwok, Benjamin; Archambault, Vincent; Topisirovic, Ivan; Tyers, Mike

Comparative small molecule screening of primary human acute leukemias, engineered human leukemia and leukemia cell lines

对原发性人类急性白血病、基因工程改造的人类白血病和白血病细胞系进行小分子药物筛选的比较研究

Safa-Tahar-Henni, Safia; Páez Martinez, Karla; Gress, Verena; Esparza, Nayeli; Roques, Élodie; Bonnet-Magnaval, Florence; Bilodeau, Mélanie; Gagné, Valérie; Bresson, Eva; Cardin, Sophie; El-Hachem, Nehme; Iasenza, Isabella; Alzial, Gabriel; Boivin, Isabel; Nakamichi, Naoto; Soufflet, Anne-Cécile; Mirela Pascariu, Cristina; Duchaine, Jean; Mathien, Simon; Bonneil, Éric; Eppert, Kolja; Marinier, Anne; Sauvageau, Guy; Deblois, Geneviève; Thibault, Pierre; Hébert, Josée; Eaves, Connie J; Cellot, Sonia; Barabé, Frédéric; Wilhelm, Brian T

DDB1 engagement defines the selectivity of S656 analogs for cyclin K degradation over CDK inhibition.

DDB1 的参与决定了 S656 类似物对细胞周期蛋白 K 降解的选择性,而非对 CDK 的抑制

Moison Céline, Mendoza-Sanchez Rodrigo, Gracias Deanne, Schuetz Doris A, Spinella Jean-François, Girard Simon, Thavonekham Bounkham, Chagraoui Jalila, Durand Aurélie, Fortier Simon, MacRae Tara, Bonneil Eric, Rose Yannick, Mayotte Nadine, Boivin Isabel, Thibault Pierre, Hébert Josée, Ruel Réjean, Marinier Anne, Sauvageau Guy

Medicinal Chemistry and NMR Driven Discovery of Novel UDP-glucuronosyltransferase 1A Inhibitors That Overcome Therapeutic Resistance in Cells

利用药物化学和核磁共振技术发现新型UDP-葡萄糖醛酸转移酶1A抑制剂,克服细胞治疗耐药性

Osborne, Michael J; Sulekha, Anamika; Culjkovic-Kraljacic, Biljana; Gasiorek, Jadwiga; Ruediger, Edward; Jolicouer, Eric; Marinier, Anne; Assouline, Sarit; Borden, Katherine L B

FRI458 Rare Pathogenic Missense Variants in LMNA Identified in Women with Polycystic Ovary Syndrome (PCOS)

在多囊卵巢综合征(PCOS)女性中发现LMNA基因的FRI458罕见致病性错义变异

Paknikar, Raghavendra; Alpert, Lindsay; Cohen, Russell D; Shogan, Benjamin; Micic, Dejan; Muralidharan, Charanya; Huiping huang, Fei; May, Sarah C; Enriquez, Jacob; Nelson, Jennifer B; Wang, Eugenia; Chakraborthy, Advaita; Figatner, Kayla T; Navitskaya, Svetlana N; Tersey, Sarah A; Mirmira, Raghavendra G; Naaman, Sandra; Sintetas, Stephanie; Van Cauter, Eve; Hanlon, Erin C; Chopra, Karishma A; Gunaratne, Naiomi C; Deplewski, Dianne; Vallet, Amandine; Diennet, Marine; Thiombane, Khady; Vivet, Anaïs; Weber, Sandra; El Ezzy, Mohamed; Shaikh, Faraz; Poupart, Julien; Mendoza-Sanchez, Rodrigo; Alexandra Schuetz, Doris; Marinier, Anne; Greene, Geoffrey L; William Fanning, Sean; Nathalie Mader, Sylvie; Rashied, Ammar; Cursio, John; Hanlon, Erin C; Pannain, Silvana; Cipriani, Nicole A; Antic, Tatjana; Banizs, Anna; Finkelstein, Sydney David; Darji, Monika; Pannain, Silvana; Sam, Susan; Van Cauter, Eve; Hanlon, Erin C; Checkcinco, Christian; Tersey, Sarah A; Mirmira, Raghavendra G; Auckley, Elizabeth Diane; Arosemena, Marilyn A; Philipson, Louis; Ettleson, Matthew D; Laiteerapong, Neda; Wan, Wen; Bianco, Antonio C; Vasavada, Sheel R; Chopra, Karishma A; Philipson, Louis; Reutrakul, Sirimon; McAnany, J Jason; Park, Jason C; Chau, Felix Y; Danielson, Kirstie K; Bharati, Prasad; Pannain, Silvana; Van Cauter, Eve; Hanlon, Erin C; Freeman, Stephen J; Radonski, Brandon; Lecka, Liam; Davis, Ka'Derricka; Prince, Grace; Carthy, Kevin; Seley, Jane J; Song, Jing; Lee, Jungwha; Bailey, Stacy C; Khorzad, Rebeca; Gatchell, David; Ankenman, Bruce; Lewis, Daniel R; Holl, Jane; Wallia, Amisha; Salas Lucia, Federico; Hui Liao, Xiao; Jiang, Hanzi; Dumitrescu, Alexandra M; Refetoff, Samuel; Anselmo, Joao; Myong, Subin; Challa, Sridevi; Desai, Jui; Letourneau-Freiberg, Lisa; Msall, Michael; Scott, Megan; Nicole Naylor, Rochelle; Philipson, Louis; Greeley, Siri Atma W; Anderson, Cara; Kulkarni, Abhishek; Maier, Bernhard; Tersey, Sarah A; Anderson, Ryan; Mirmira, Raghavendra G; Ermis, Ebru; Nargis, Titli; Kulkarni, Abhishek; May, Sarah; Tersey, Sarah A; Mirmira, Raghavendra G; Anderson, Ryan M; Webster, Kierstin L; Wu, Wenting; Webb-Robertson, Bobbie-Jo; Nakayasu, Ernesto; Sarkar, Soumyadeep; Evans-Molina, Carmella; Tersey, Sarah A; Enriquez, Jacob; Hammes, Stephen R; Mirmira, Raghavendra G; Yang, Qiwei; Al-Hendy, Ayman; Bullock, Cydney A; Davis, Ka'Derricka; Carthy, Kevin; Wax, Pamela; Smyrniotis, Colleen; Pollack, Teresa; Barnard, Cynthia; Holl, Jane; Wallia, Amisha; Hammoud, Batoul; DiMeglio, Linda A; Kulkarni, Abishek; Hull, Audrey; Woerner, Stephanie; Cabrera, Susanne; Mastrandrea, Lucy D; Ouyang, Fangian; Perkins, Susan N; Evans-Molina, Carmella; Mastracci, Teresa L; Tersey, Sarah A; Sarkar, Soumyaddep; Nakayasu, Ernesto; Webb-Robertson, Bobbie-Jo; Gerner, Eugene; Mirmira, Raghavendra G; Sims, Emily K; Clarke, Bart; Aziz Khan, Aliya; Ruth Rubin, Mishaela; Schwarz, Peter E; Vokes, Tamara J; Shoback, Dolores M; Gagnon, Claudia; Palermo, Andrea; Abbott, Lisa G; Hofbauer, Lorenz C; Kohlmeier, Lynn; Cetani, Filomena; Phil, Susanne; An, Xuebei; Raymond Smith, Alden; Lai, Bryant; Le, John; Ukena, Jenny; Sibley, Christopher; Shu, Aimee; Rejnmark, Lars; Hancock, Govinda; Young, Kristen; Greene, Geoffrey L; Fanning, Sean William; Arosemena, Marilyn A; Wroblewski, Kristen; Tasali, Esra; Philipson, Louis H; Baboun, Daniela; Solano, Natalia; Sanchez, Andrea Martinez; Brathwaite, Carole; Restrepo, Ricardo; Alkhoury, Fuad; Carrillo-Iregui, Adriana; Li, Yanliang; Danielson, Kirstie K; Changhum Park, Jason; McAnany, J Jason; Chau, Felix Y; Prasad, Bharati; Hanlon, Erin C; Reutrakul, Sirimon; Salas Lucia, Federico; Dumitrescu, Alexandra M; Refetoff, Samuel; huang, fei; Nelson, Jennifer; Muralidharan, Charanya; Nakayasu, Ernesto; Yi, Xiaoyan; Eizirik, Decio; May, Sarah; Tersey, Sarah A; Mirmira, Raghavendra G; Nargis, Titli; Chakraborty, Advaita; Figatner, Kayla; Maloney, David; Boxer, Matthew; Tersey, Sarah A; Mirmira, Raghavendra G; Sidhu, Gurmanpreet; Madahar, Inderpreet; Haider, Adnan; Giordano, Jennifer; Liu, Jannel; Angelos, Peter; Barhoum, Maan; Jain, Rajesh; Kim, Keun Young; Hwang, Jessica; Sam, Susan; Bauer, Rosemary; Gorsic, Lidija; Legro, Richard S; Ehrmann, David; Geoffrey Hayes, M; Urbanek, Margrit

Vesicular trafficking is a key determinant of the statin response in acute myeloid leukemia

囊泡运输是急性髓系白血病中他汀类药物反应的关键决定因素。

Krosl, Jana; Bordeleau, Marie-Eve; Moison, Céline; MacRae, Tara; Boivin, Isabel; Mayotte, Nadine; Gracias, Deanne; Baccelli, Irène; Lavallée, Vincent-Philippe; Bisaillon, Richard; Lehnertz, Bernhard; Mendoza-Sanchez, Rodrigo; Ruel, Réjean; Bertomeu, Thierry; Coulombe-Huntington, Jasmin; Boucher, Geneviève; Noronha, Nandita; Pabst, Caroline; Tyers, Mike; Gendron, Patrick; Lemieux, Sébastien; Barabé, Frédéric; Marinier, Anne; Hébert, Josée; Sauvageau, Guy

Dual-Target Inhibitors of the Folate Pathway Inhibit Intrinsically Trimethoprim-Resistant DfrB Dihydrofolate Reductases

叶酸通路双靶点抑制剂抑制固有耐甲氧苄啶的DfrB二氢叶酸还原酶

Toulouse, Jacynthe L; Shi, Genbin; Lemay-St-Denis, Claudèle; Ebert, Maximilian C C J C; Deon, Daniel; Gagnon, Marc; Ruediger, Edward; Saint-Jacques, Kévin; Forge, Delphine; Vanden Eynde, Jean Jacques; Marinier, Anne; Ji, Xinhua; Pelletier, Joelle N

Complex karyotype AML displays G2/M signature and hypersensitivity to PLK1 inhibition

复杂核型急性髓系白血病表现出G2/M期特征和对PLK1抑制剂的超敏反应

Moison, Céline; Lavallée, Vincent-Philippe; Thiollier, Clarisse; Lehnertz, Bernhard; Boivin, Isabel; Mayotte, Nadine; Gareau, Yves; Fréchette, Mélanie; Blouin-Chagnon, Valérie; Corneau, Sophie; Lavallée, Sylvie; Lemieux, Sébastien; Marinier, Anne; Hébert, Josée; Sauvageau, Guy

Enhancing the drug discovery process: Bayesian inference for the analysis and comparison of dose-response experiments

增强药物发现过程:利用贝叶斯推断分析和比较剂量反应实验

Labelle, Caroline; Marinier, Anne; Lemieux, Sébastien

High-throughput screening in niche-based assay identifies compounds to target preleukemic stem cells

基于微环境的高通量筛选可鉴定靶向白血病前期干细胞的化合物

Gerby, Bastien; Veiga, Diogo F T; Krosl, Jana; Nourreddine, Sami; Ouellette, Julianne; Haman, André; Lavoie, Geneviève; Fares, Iman; Tremblay, Mathieu; Litalien, Véronique; Ottoni, Elizabeth; Kosic, Milena; Geoffrion, Dominique; Ryan, Joël; Maddox, Paul S; Chagraoui, Jalila; Marinier, Anne; Hébert, Josée; Sauvageau, Guy; Kwok, Benjamin H; Roux, Philippe P; Hoang, Trang