A-887826 is a structurally novel, potent and voltage-dependent Na(v)1.8 sodium channel blocker that attenuates neuropathic tactile allodynia in rats
A-887826 是一种结构新颖、有效且电压依赖性的 Na(v)1.8 钠通道阻滞剂,可减轻大鼠的神经性触觉异常性疼痛
期刊:Neuropharmacology
影响因子:4.6
doi:10.1016/j.neuropharm.2010.05.009
Xu-Feng Zhang, Char-Chang Shieh, Mark L Chapman, Mark A Matulenko, Ahmed H Hakeem, Robert N Atkinson, Michael E Kort, Brian E Marron, Shailen Joshi, Prisca Honore, Connie R Faltynek, Douglas S Krafte, Michael F Jarvis