日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Cryptosporidium PI(4)K inhibitor EDI048 is a gut-restricted parasiticidal agent to treat paediatric enteric cryptosporidiosis

隐孢子虫 PI(4)K 抑制剂 EDI048 是一种肠道限制性杀寄生虫剂,用于治疗儿童肠道隐孢子虫病

Ujjini H Manjunatha #, Suresh B Lakshminarayana #, Rajiv S Jumani #, Alexander T Chao, Joseph M Young, Jonathan E Gable, Mark Knapp, Imad Hanna, Jean-Rene Galarneau, John Cantwell, Upendra Kulkarni, Michael Turner, Peichao Lu, Kristen H Darrell, Lucy C Watson, Katherine Chan, Debjani Patra, Mulugeta

Impact of COVID-19 pandemic on depression incidence and healthcare service use among patients with depression: an interrupted time-series analysis from a 9-year population-based study

COVID-19 大流行对抑郁症发病率和抑郁症患者医疗保健服务利用的影响:一项基于 9 年人群研究的中断时间序列分析

Chan, Vivien Kin Yi; Chai, Yi; Chan, Sandra Sau Man; Luo, Hao; Jit, Mark; Knapp, Martin; Bishai, David Makram; Ni, Michael Yuxuan; Wong, Ian Chi Kei; Li, Xue

Identification of Potent, Broad-Spectrum Coronavirus Main Protease Inhibitors for Pandemic Preparedness

为应对大流行而鉴定高效广谱冠状病毒主蛋白酶抑制剂

David T Barkan ,Keira Garland ,Lei Zhang ,Richard T Eastman ,Matthew Hesse ,Mark Knapp ,Elizabeth Ornelas ,Jenny Tang ,Wilian Augusto Cortopassi ,Yu Wang ,Frederick King ,Weiping Jia ,Zachary Nguyen ,Andreas O Frank ,Ryan Chan ,Eric Fang ,Daniel Fuller ,Scott Busby ,Heidi Carias ,Kristine Donahue ,Laura Tandeske ,Thierry T Diagana ,Nadine Jarrousse ,Heinz Moser ,Christopher Sarko ,Dustin Dovala ,Stephanie Moquin ,Vanessa M Marx

mRNA Display Identifies Potent, Paralog-Selective Peptidic Ligands for ARID1B

mRNA 显示可识别 ARID1B 的有效、旁系同源选择性肽配体

Gregor S Cremosnik, Yannick Mesrouze, Patrik Zueger, David Furkert, Frédéric Grandjean, Dayana Argoti, Fanny Mermet-Meillon, Matthias R Bauer, Scott Brittain, Phuong Rogemoser, Winnie Yang, Jerome Giovannoni, Lynn McGregor, Jenny Tang, Mark Knapp, Sandra Holzinger, Sylvia Buhr, Lionel Muller, Lukas

Structural basis of indisulam-mediated RBM39 recruitment to DCAF15 E3 ligase complex

吲哚磺胺介导的 RBM39 募集至 DCAF15 E3 连接酶复合物的结构基础

Dirksen E Bussiere, Lili Xie, Honnappa Srinivas, Wei Shu, Ashley Burke, Celine Be, Junping Zhao, Adarsh Godbole, Dan King, Rajeshri G Karki, Viktor Hornak, Fangmin Xu, Jennifer Cobb, Nathalie Carte, Andreas O Frank, Alexandra Frommlet, Patrick Graff, Mark Knapp, Aleem Fazal, Barun Okram, Songchun Ji

A polyomavirus peptide binds to the capsid VP1 pore and has potent antiviral activity against BK and JC polyomaviruses

多瘤病毒肽与衣壳 VP1 孔结合,对 BK 和 JC 多瘤病毒具有强效抗病毒活性

Joshua R Kane, Susan Fong, Jacob Shaul, Alexandra Frommlet, Andreas O Frank, Mark Knapp, Dirksen E Bussiere, Peter Kim, Elizabeth Ornelas, Carlos Cuellar, Anastasia Hyrina, Johanna R Abend, Charles A Wartchow