日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Targeting HIF-activated collagen prolyl 4-hydroxylase expression disrupts collagen deposition and blocks primary and metastatic uveal melanoma growth

靶向 HIF 激活的胶原脯氨酰 4-羟化酶表达可破坏胶原沉积并阻止原发性和转移性葡萄膜黑色素瘤的生长

Stefan Kaluz #, Qing Zhang #, Yuki Kuranaga, Hua Yang, Satoru Osuka, Debanjan Bhattacharya, Narra S Devi, Jiyoung Mun, Wei Wang, Ruiwen Zhang, Mark M Goodman, Hans E Grossniklaus, Erwin G Van Meir

A Swine Hind Limb Ischemia Model Useful for Testing Peripheral Artery Disease Therapeutics

用于测试外周动脉疾病治疗的猪后肢缺血模型

Juline N Deppen, Sydney C Ginn, Na Hee Kim, Lanfang Wang, Ronald J Voll, Steven H Liang, Mark M Goodman, John N Oshinski, Rebecca D Levit

PET Tracer 18F-Fluciclovine Can Detect Histologically Proven Bone Metastatic Lesions: A Preclinical Study in Rat Osteolytic and Osteoblastic Bone Metastasis Models

PET 示踪剂 18F-氟西洛维可检测出经组织学证实的骨转移病变:大鼠溶骨性和成骨性骨转移模型中的临床前研究

Shuntaro Oka, Masaru Kanagawa, Yoshihiro Doi, David M Schuster, Mark M Goodman, Hirokatsu Yoshimura

[(14)C]Fluciclovine (alias anti-[(14)C]FACBC) uptake and ASCT2 expression in castration-resistant prostate cancer cells

去势抵抗性前列腺癌细胞中[(14)C]氟西氯维因(别名抗-[(14)C]FACBC)的摄取和ASCT2的表达

Masahiro Ono, Shuntaro Oka, Hiroyuki Okudaira, Takeo Nakanishi, Atsushi Mizokami, Masato Kobayashi, David M Schuster, Mark M Goodman, Yoshifumi Shirakami, Keiichi Kawai

Design and in vitro activities of N-alkyl-N-[(8-R-2,2-dimethyl-2H-chromen-6-yl)methyl]heteroarylsulfonamides, novel, small-molecule hypoxia inducible factor-1 pathway inhibitors and anticancer agents

N-烷基-N-[(8-R-2,2-二甲基-2H-色满-6-基)甲基]杂芳基磺酰胺、新型小分子缺氧诱导因子-1通路抑制剂和抗癌剂的设计和体外活性

Jiyoung Mun, Adnan Abdul Jabbar, Narra Sarojini Devi, Shaoman Yin, Yingzhe Wang, Chalet Tan, Deborah Culver, James P Snyder, Erwin G Van Meir, Mark M Goodman

Binding Model for the Interaction of Anticancer Arylsulfonamides with the p300 Transcription Cofactor

抗癌芳基磺酰胺与 p300 转录辅因子相互作用的结合模型

Qi Shi, Shaoman Yin, Stefan Kaluz, Nanting Ni, Narra Sarojini Devi, Jiyoung Mun, Danzhu Wang, Krishna Damera, Weixuan Chen, Sarah Burroughs, Suazette Reid Mooring, Mark M Goodman, Erwin G Van Meir, Binghe Wang, James P Snyder