日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Synthesis of vancomycin fluorescent probes that retain antimicrobial activity, identify Gram-positive bacteria, and detect Gram-negative outer membrane damage

保留抗菌活性、识别革兰氏阳性菌、检测革兰氏阴性外膜损伤的万古霉素荧光探针的合成

Bing Zhang, Wanida Phetsang, M Rhia L Stone, Sanjaya Kc, Mark S Butler, Matthew A Cooper, Alysha G Elliott, Urszula Łapińska, Margaritis Voliotis, Krasimira Tsaneva-Atanasova, Stefano Pagliara, Mark A T Blaskovich

An amphipathic peptide with antibiotic activity against multidrug-resistant Gram-negative bacteria

具有针对多重耐药革兰氏阴性细菌的抗生素活性的两亲肽

Alysha G Elliott #, Johnny X Huang #, Søren Neve, Johannes Zuegg, Ingrid A Edwards, Amy K Cain, Christine J Boinett, Lars Barquist, Carina Vingsbo Lundberg, Jason Steen, Mark S Butler, Mehdi Mobli, Kaela M Porter, Mark A T Blaskovich, Sergio Lociuro, Magnus Strandh, Matthew A Cooper

Octapeptin C4 and polymyxin resistance occur via distinct pathways in an epidemic XDR Klebsiella pneumoniae ST258 isolate

流行性 XDR 肺炎克雷伯菌 ST258 分离株通过不同途径发生八肽霉素 C4 和多粘菌素耐药性

Miranda E Pitt, Minh Duc Cao, Mark S Butler, Soumya Ramu, Devika Ganesamoorthy, Mark A T Blaskovich, Lachlan J M Coin, Matthew A Cooper

Protein-inspired antibiotics active against vancomycin- and daptomycin-resistant bacteria

蛋白质启发抗生素可有效对抗万古霉素和达托霉素耐药细菌

Mark A T Blaskovich, Karl A Hansford, Yujing Gong, Mark S Butler, Craig Muldoon, Johnny X Huang, Soumya Ramu, Alberto B Silva, Mu Cheng, Angela M Kavanagh, Zyta Ziora, Rajaratnam Premraj, Fredrik Lindahl, Tanya A Bradford, June C Lee, Tomislav Karoli, Ruby Pelingon, David J Edwards, Maite Amado, Aly

Design, Synthesis, and Biological Evaluation of 2-Nitroimidazopyrazin-one/-es with Antitubercular and Antiparasitic Activity

具有抗结核和抗寄生虫活性的 2-硝基咪唑并吡嗪酮的设计、合成及生物学评价

Angie M Jarrad, Chee Wei Ang, Anjan Debnath, Hye Jee Hahn, Kyra Woods, Lendl Tan, Melissa L Sykes, Amy J Jones, Ruby Pelingon, Mark S Butler, Vicky M Avery, Nicholas P West, Tomislav Karoli, Mark A T Blaskovich, Matthew A Cooper

Structure, Function, and Biosynthetic Origin of Octapeptin Antibiotics Active against Extensively Drug-Resistant Gram-Negative Bacteria

八肽素抗生素的结构、功能和生物合成来源,可有效对抗广泛耐药的革兰氏阴性细菌

Tony Velkov, Alejandra Gallardo-Godoy, James D Swarbrick, Mark A T Blaskovich, Alysha G Elliott, Meiling Han, Philip E Thompson, Kade D Roberts, Johnny X Huang, Bernd Becker, Mark S Butler, Lawrence H Lash, Sónia Troeira Henriques, Roger L Nation, Sivashangarie Sivanesan, Marc-Antoine Sani, Frances

Pharmacological targeting of the transcription factor SOX18 delays breast cancer in mice

转录因子 SOX18 的药理靶向作用可延缓小鼠乳腺癌

Jeroen Overman, Frank Fontaine #, Mehdi Moustaqil #, Deepak Mittal, Emma Sierecki, Natalia Sacilotto, Johannes Zuegg, Avril A B Robertson, Kelly Holmes, Angela A Salim, Sreeman Mamidyala, Mark S Butler, Ashley S Robinson, Emmanuelle Lesieur, Wayne Johnston, Kirill Alexandrov, Brian L Black, Benjamin

Fluorescent Trimethoprim Conjugate Probes To Assess Drug Accumulation in Wild Type and Mutant Escherichia coli

荧光甲氧苄啶结合探针评估野生型和突变型大肠杆菌中的药物积累

Wanida Phetsang, Ruby Pelingon, Mark S Butler, Sanjaya Kc, Miranda E Pitt, Geraldine Kaeslin, Matthew A Cooper, Mark A T Blaskovich

A small-molecule inhibitor of the NLRP3 inflammasome for the treatment of inflammatory diseases

NLRP3炎症小体的小分子抑制剂用于治疗炎症疾病

Rebecca C Coll, Avril A B Robertson, Jae Jin Chae, Sarah C Higgins, Raúl Muñoz-Planillo, Marco C Inserra, Irina Vetter, Lara S Dungan, Brian G Monks, Andrea Stutz, Daniel E Croker, Mark S Butler, Moritz Haneklaus, Caroline E Sutton, Gabriel Núñez, Eicke Latz, Daniel L Kastner, Kingston H G Mills, Se

Mucin Binding Reduces Colistin Antimicrobial Activity

粘蛋白结合降低粘菌素抗菌活性

Johnny X Huang, Mark A T Blaskovich, Ruby Pelingon, Soumya Ramu, Angela Kavanagh, Alysha G Elliott, Mark S Butler, A Bruce Montgomery, Matthew A Cooper