日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

UBE2N Is Essential for Maintenance of Skin Homeostasis and Suppression of Inflammation

UBE2N对于维持皮肤稳态和抑制炎症至关重要

Lee, Min Jin; Hammouda, Manel Ben; Miao, Wanying; Okafor, Arinze E; Jin, Yingai J; Sun, Huiying; Jain, Vaibhav; Markovtsov, Vadim; Diao, Yarui; Gregory, Simon G; Zhang, Jennifer Y

UBE2N is essential for maintenance of skin homeostasis and suppression of inflammation

UBE2N 对于维持皮肤稳态和抑制炎症至关重要

Min Jin Lee, Manel Ben Hammouda, Wanying Miao, Arinze Okafor, Yingai Jin, Huiying Sun, Vaibhav Jain, Vadim Markovtsov, Yarui Diao, Simon G Gregory, Jennifer Y Zhang

Assessment of thrombotic risk during long-term treatment of immune thrombocytopenia with fostamatinib

使用福斯他替尼长期治疗免疫性血小板减少症期间的血栓风险评估

Cooper, Nichola; Altomare, Ivy; Thomas, Mark R; Nicolson, Phillip L R; Watson, Steve P; Markovtsov, Vadim; Todd, Leslie K; Masuda, Esteban; Bussel, James B

Fostamatinib for the treatment of adult persistent and chronic immune thrombocytopenia: Results of two phase 3, randomized, placebo-controlled trials

福斯他替尼治疗成人持续性和慢性免疫性血小板减少症:两项 3 期随机、安慰剂对照试验的结果

Bussel, James; Arnold, Donald M; Grossbard, Elliot; Mayer, Jiří; Treliński, Jacek; Homenda, Wojciech; Hellmann, Andrzej; Windyga, Jerzy; Sivcheva, Liliya; Khalafallah, Alhossain A; Zaja, Francesco; Cooper, Nichola; Markovtsov, Vadim; Zayed, Hany; Duliege, Anne-Marie

1364. Efficacy of Omadacycline Against Molecularly Characterized Gram-Positive and Gram-Negative Pathogens Causing Infections in the Phase 3 CABP and ABSSSI Clinical Trials

1364. 奥马环素对分子鉴定的革兰氏阳性菌和革兰氏阴性菌感染的疗效(在3期社区获得性细菌性肺炎和急性细菌性皮肤及皮肤结构感染临床试验中)

Kruć-Fijałkowska, Roksana; Drożdżyński, Dariusz; Matusiak, Magdalena; Dragon, Krzysztof; Szczepański, Marek; Gotur, Deepa B; Malik, Anuj; Markovtsov, Vadim; Yan, Lucy; Dummer, Wolfgang; Mallat, Ziad; Mendes, Rodrigo E; Castanheira, Mariana; Armstrong, Eliana S; Steenbergen, Judith N; Flamm, Robert K

Exercise performance and peripheral vascular insufficiency improve with AMPK activation in high-fat diet-fed mice

高脂饮食喂养的小鼠的运动表现和外周血管功能不全随着 AMPK 激活而改善

Kristen A Baltgalvis, Kathy White, Wei Li, Mark D Claypool, Wayne Lang, Raniel Alcantara, Baljit K Singh, Annabelle M Friera, John McLaughlin, Derek Hansen, Kelly McCaughey, Henry Nguyen, Ira J Smith, Guillermo Godinez, Simon J Shaw, Dane Goff, Rajinder Singh, Vadim Markovtsov, Tian-Qiang Sun, Yonch

Global metabolite profiling of mice with high-fat diet-induced obesity chronically treated with AMPK activators R118 or metformin reveals tissue-selective alterations in metabolic pathways

对高脂饮食诱导肥胖的小鼠进行全球代谢物分析,并长期使用 AMPK 激活剂 R118 或二甲双胍进行治疗,结果显示代谢途径存在组织选择性改变。

Jenkins, Yonchu; Sun, Tian-Qiang; Li, Yingwu; Markovtsov, Vadim; Uy, Gerald; Gross, Lisa; Goff, Dane A; Shaw, Simon J; Boralsky, Luke; Singh, Rajinder; Payan, Donald G; Hitoshi, Yasumichi

AMPK activation through mitochondrial regulation results in increased substrate oxidation and improved metabolic parameters in models of diabetes

通过线粒体调节激活 AMPK 可增加底物氧化并改善糖尿病模型中的代谢参数

Yonchu Jenkins, Tian-Qiang Sun, Vadim Markovtsov, Marc Foretz, Wei Li, Henry Nguyen, Yingwu Li, Alison Pan, Gerald Uy, Lisa Gross, Kristen Baltgalvis, Stephanie L Yung, Tarikere Gururaja, Taisei Kinoshita, Alexander Owyang, Ira J Smith, Kelly McCaughey, Kathy White, Guillermo Godinez, Raniel Alcanta

Preclinical characterization of Aurora kinase inhibitor R763/AS703569 identified through an image-based phenotypic screen.

通过基于图像的表型筛选鉴定的 Aurora 激酶抑制剂 R763/AS703569 的临床前表征

McLaughlin John, Markovtsov Vadim, Li Hui, Wong Steve, Gelman Marina, Zhu Yanhong, Franci Christian, Lang D Wayne, Pali Erlina, Lasaga Joe, Low Caroline, Zhao Feifei, Chang Betty, Gururaja Tarikere L, Xu Weiduan, Baluom Muhammad, Sweeny David, Carroll David, Sran Arvinder, Thota Sambaiah, Parmer Manjeet, Romane Angela, Clemens George, Grossbard Elliott, Qu Kunbin, Jenkins Yonchu, Kinoshita Taisei, Taylor Vanessa, Holland Sacha J, Argade Ankush, Singh Rajinder, Pine Polly, Payan Donald G, Hitoshi Yasumichi

Critical role of the ubiquitin ligase activity of UHRF1, a nuclear RING finger protein, in tumor cell growth

UHRF1(一种核内RING指蛋白)的泛素连接酶活性在肿瘤细胞生长中起着关键作用

Jenkins, Yonchu; Markovtsov, Vadim; Lang, Wayne; Sharma, Poonam; Pearsall, Denise; Warner, Justin; Franci, Christian; Huang, Betty; Huang, Jianing; Yam, George C; Vistan, Joseph P; Pali, Erlina; Vialard, Jorge; Janicot, Michel; Lorens, James B; Payan, Donald G; Hitoshi, Yasumichi