日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Formulation and Evaluation of Alginate Microcapsules Containing an Uncompetitive Nanomolar Dimeric Indenoindole Inhibitor of the Human Breast Cancer Resistance Pump ABCG2 with Different Excipients

配制和评价含有非竞争性纳摩尔级二聚体茚并吲哚类化合物(人乳腺癌耐药泵ABCG2抑制剂)的藻酸盐微胶囊及其不同赋形剂

Bodnár, Krisztina; Marminon, Christelle; Perret, Florent; Haimhoffer, Ádám; Papp, Boglárka; Fehér, Pálma; Ujhelyi, Zoltán; Jose, Joachim; Le Borgne, Marc; Bácskay, Ildikó; Józsa, Liza

Formulation and Investigation of CK2 Inhibitor-Loaded Alginate Microbeads with Different Excipients

制备和研究含不同辅料的CK2抑制剂藻酸盐微球

Papp, Boglárka; Le Borgne, Marc; Perret, Florent; Marminon, Christelle; Józsa, Liza; Pető, Ágota; Kósa, Dóra; Nagy, Lajos; Kéki, Sándor; Ujhelyi, Zoltán; Pallér, Ádám; Budai, István; Bácskay, Ildikó; Fehér, Pálma

Synthesis, in silico study (DFT, ADMET) and crystal structure of novel sulfamoyloxy-oxazolidinones: Interaction with SARS-CoV-2

新型磺酰氧基噁唑烷酮的合成、计算机模拟研究(DFT、ADMET)和晶体结构:与SARS-CoV-2的相互作用

Bouzina, Abdeslem; Berredjem, Malika; Bouacida, Sofiane; Bachari, Khaldoun; Marminon, Christelle; Borgne, Marc Le; Bouaziz, Zouhair; Bouone, Yousra Ouafa

Broad-Spectrum Anticancer Activity and Pharmacokinetic Properties of a Prenyloxy-Substituted Indeno[1,2-b]indole Derivative, Discovered as CK2 Inhibitor

一种异戊烯氧基取代的茚并[1,2-b]吲哚衍生物的广谱抗癌活性和药代动力学特性,该衍生物被发现是CK2抑制剂

El-Awaad, Ehab; Birus, Robin; Marminon, Christelle; Bouaziz, Zouhair; Ballentin, Laurens; Aichele, Dagmar; Le Borgne, Marc; Jose, Joachim

Mechanistic basis of breast cancer resistance protein inhibition by new indeno[1,2-b]indoles

新型茚并[1,2-b]吲哚抑制乳腺癌耐药蛋白的机制基础

Diogo Henrique Kita #, Nathalie Guragossian #, Ingrid Fatima Zattoni, Vivian Rotuno Moure, Fabiane Gomes de Moraes Rego, Sabrina Lusvarghi, Thomas Moulenat, Billel Belhani, Geraldo Picheth, Sofiane Bouacida, Zouhair Bouaziz, Christelle Marminon, Malika Berredjem, Joachim Jose, Marcos Brown Gonçalves

Diacritic Binding of an Indenoindole Inhibitor by CK2α Paralogs Explored by a Reliable Path to Atomic Resolution CK2α' Structures

通过可靠的原子分辨率CK2α'结构解析方法探索CK2α旁系同源物对茚并吲哚抑制剂的重音符号结合

Lindenblatt, Dirk; Nickelsen, Anna; Applegate, Violetta M; Hochscherf, Jennifer; Witulski, Benedict; Bouaziz, Zouhair; Marminon, Christelle; Bretner, Maria; Le Borgne, Marc; Jose, Joachim; Niefind, Karsten

QSAR Model of Indeno[1,2- b]indole Derivatives and Identification of N-isopentyl-2-methyl-4,9-dioxo-4,9-Dihydronaphtho[2,3- b]furan-3-carboxamide as a Potent CK2 Inhibitor

茚并[1,2- b]吲哚衍生物的 QSAR 模型以及 N-异戊基-2-甲基-4,9-二氧代-4,9-二氢萘并[2,3- b]呋喃-3-甲酰胺作为强效 CK2 抑制剂的鉴定

Samer Haidar, Christelle Marminon, Dagmar Aichele, Abdelhamid Nacereddine, Wael Zeinyeh, Abdeslem Bouzina, Malika Berredjem, Laurent Ettouati, Zouhair Bouaziz, Marc Le Borgne, Joachim Jose

Inhibition of Shiga toxin-converting bacteriophage development by novel antioxidant compounds

新型抗氧化化合物抑制志贺毒素转化噬菌体的发育

Sylwia Bloch, Bożena Nejman-Faleńczyk, Karolina Pierzynowska, Ewa Piotrowska, Alicja Węgrzyn, Christelle Marminon, Zouhair Bouaziz, Pascal Nebois, Joachim Jose, Marc Le Borgne, Luciano Saso, Grzegorz Węgrzyn

Self-Assembled Supramolecular Nanoparticles Improve the Cytotoxic Efficacy of CK2 Inhibitor THN7

自组装超分子纳米粒子提高了CK2抑制剂THN7的细胞毒性功效

Nacereddine, Abdelhamid; Bollacke, Andre; Róka, Eszter; Marminon, Christelle; Bouaziz, Zouhair; Fenyvesi, Ferenc; Bácskay, Ildikó Katalin; Jose, Joachim; Perret, Florent; Le Borgne, Marc

Development of Pharmacophore Model for Indeno[1,2-b]indoles as Human Protein Kinase CK2 Inhibitors and Database Mining

构建吲哚并[1,2-b]吲哚类化合物作为人蛋白激酶CK2抑制剂的药效团模型及数据库挖掘

Haidar, Samer; Bouaziz, Zouhair; Marminon, Christelle; Laitinen, Tuomo; Poso, Antti; Le Borgne, Marc; Jose, Joachim