日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Discovery, Structure-Activity Relationship, and Functional Characterization of a Chromenopyrrole Series as Orthosteric Antagonists of GPR84

色烯吡咯系列化合物作为GPR84正构拮抗剂的发现、构效关系及功能表征

Malone, Michael A; Yin, Ruijing; Li, Yueming; Jenkins, Laura; Guseinov, Abdul-Akim; Marsango, Sara; Huggett, Mark; Huggett, Margaret; Boyle, Anna; Morrison, Angus; Tikhonova, Irina G; Milligan, Graeme; Jamieson, Andrew G

Allosteric modulation and biased signalling at free fatty acid receptor 2

游离脂肪酸受体 2 的变构调节和偏向性信号传导

Zhang, Xuan; Guseinov, Abdul-Akim; Jenkins, Laura; Valentini, Alice; Marsango, Sara; Schultz-Knudsen, Katrine; Ulven, Trond; Rexen Ulven, Elisabeth; Tikhonova, Irina G; Milligan, Graeme; Zhang, Cheng

Steric control of signaling bias in the immunometabolic receptor GPR84

免疫代谢受体 GPR84 中信号偏向的空间控制

Wang, Pinqi; Zhang, Xuan; Guseinov, Abdul-Akim; Jenkins, Laura; von Hallerstein, Carl; Colburn, Jonathan D; Ives, Rowan; Luscombe, Vincent B; Marsango, Sara; Oktavia, Listiana; Raja, Arun; Greaves, David R; Biggin, Philip C; Milligan, Graeme; Zhang, Cheng; Tikhonova, Irina G; Russell, Angela J

PET Imaging of Innate Immune Activation Using 11C Radiotracers Targeting GPR84

使用 11C 放射性示踪剂靶向 GPR84 进行先天免疫激活的 PET 成像

Mausam Kalita, Jun Hyung Park, Renesmee Chenting Kuo, Samira Hayee, Sara Marsango, Valentina Straniero, Israt S Alam, Angelie Rivera-Rodriguez, Mallesh Pandrala, Mackenzie L Carlson, Samantha T Reyes, Isaac M Jackson, Lorenzo Suigo, Audrey Luo, Sydney C Nagy, Ermanno Valoti, Graeme Milligan, Frezghi

Phosphorylation bar-coding of free fatty acid receptor 2 is generated in a tissue-specific manner

游离脂肪酸受体 2 的磷酸化条形码以组织特异性方式产生

Natasja Barki, Laura Jenkins, Sara Marsango, Domonkos Dedeo, Daniele Bolognini, Louis Dwomoh, Aisha M Abdelmalik, Margaret Nilsen, Manon Stoffels, Falko Nagel, Stefan Schulz, Andrew B Tobin, Graeme Milligan

Therapeutic validation of an orphan G protein-coupled receptor: The case of GPR84

孤儿G蛋白偶联受体的治疗验证:以GPR84为例

Marsango, Sara; Barki, Natasja; Jenkins, Laura; Tobin, Andrew B; Milligan, Graeme

LBODP079 A Case of Silent Invasive Corticotroph Adenoma

LBODP079 一例无症状侵袭性促肾上腺皮质激素腺瘤

Brown, C H; Bains, J S; Ludwig, M; Stern, J E; Marsango, Sara; Bonaccorsi di Patti, Maria Carmela; Barra, Donatella; Miele, Rossella; Azmath, Misbath; Faisal, Sobia; Kantorovich, Vitaly; Guruli, Marie; Bendaram, Snigdha Reddy; Kantorovich, Vitaly

Selective phosphorylation of threonine residues defines GPR84-arrestin interactions of biased ligands

苏氨酸残基的选择性磷酸化决定了偏向配体的 GPR84-arrestin 相互作用

Sara Marsango, Richard J Ward, Laura Jenkins, Adrian J Butcher, Zobaer Al Mahmud, Louis Dwomoh, Falko Nagel, Stefan Schulz, Irina G Tikhonova, Andrew B Tobin, Graeme Milligan

The M1 muscarinic receptor is present in situ as a ligand-regulated mixture of monomers and oligomeric complexes

M1 毒蕈碱受体以配体调节的单体和寡聚复合物混合物的形式存在

Sara Marsango, Laura Jenkins, John D Pediani, Sophie J Bradley, Richard J Ward, Sarah Hesse, Gabriel Biener, Michael R Stoneman, Andrew B Tobin, Valerica Raicu, Graeme Milligan

Biased M1 muscarinic receptor mutant mice show accelerated progression of prion neurodegenerative disease

M1毒蕈碱受体偏向性突变小鼠表现出朊病毒神经退行性疾病进展加速。

Scarpa, Miriam; Molloy, Colin; Jenkins, Laura; Strellis, Bethany; Budgett, Rebecca F; Hesse, Sarah; Dwomoh, Louis; Marsango, Sara; Tejeda, Gonzalo S; Rossi, Mario; Ahmed, Zeshan; Milligan, Graeme; Hudson, Brian D; Tobin, Andrew B; Bradley, Sophie J