日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Targeting CCNE1 amplified ovarian and endometrial cancers by combined inhibition of PKMYT1 and ATR

通过联合抑制PKMYT1和ATR靶向CCNE1扩增的卵巢癌和子宫内膜癌

Xu, Haineng; George, Erin; Gallo, David; Medvedev, Sergey; Wang, Xiaolei; Datta, Arindam; Kryczka, Rosie; Hyer, Marc L; Fourtounis, Jimmy; Stocco, Rino; Aguado-Fraile, Elia; Petrone, Adam; Yin, Shou Yun; Shiwram, Ariya; Liu, Fang; Anderson, Matthew; Kim, Hyoung; Greenberg, Roger A; Marshall, C Gary; Simpkins, Fiona

PKMYT1 inhibition induces DNA damage and synergizes with immune checkpoint blockade in CCNE1 -amplified gastroesophageal adenocarcinoma

PKMYT1抑制可诱导DNA损伤,并与CCNE1扩增的胃食管腺癌中的免疫检查点阻断产生协同作用。

Jang, Sungjoo; Wu, Lawrence W; Park, Jimyung; Hangai, Sho; Shapiro, Cameron; Marshall, C Gary; Cai, Luke L; Izar, Benjamin; Bass, Adam J; Moy, Ryan H

Low-Molecular Weight Cyclin E Confers a Vulnerability to PKMYT1 Inhibition in Triple-Negative Breast Cancer.

低分子量细胞周期蛋白 E 使三阴性乳腺癌对 PKMYT1 抑制剂敏感

Li Mi, Lulla Amriti R, Wang Yan, Tsavaschidis Spyros, Wang Fuchenchu, Karakas Cansu, Nguyen Tuyen D T, Bui Tuyen N, Pina Marc A, Chen Mei-Kuang, Mastoraki Sofia, Multani Asha S, Fowlkes Natalie W, Sahin Aysegul, Marshall C Gary, Hunt Kelly K, Keyomarsi Khandan

HDAC11 deficiency disrupts oncogene-induced hematopoiesis in myeloproliferative neoplasms

HDAC11 缺陷会破坏骨髓增生性肿瘤中癌基因诱导的造血作用

Yue, Lanzhu; Sharma, Vasundhara; Horvat, Nathan P; Akuffo, Afua A; Beatty, Matthew S; Murdun, Cem; Colin, Christelle; Billington, Julia M R; Goodheart, William E; Sahakian, Eva; Zhang, Ling; Powers, John J; Amin, Narmin E; Lambert-Showers, Que T; Darville, Lancia N; Pinilla-Ibarz, Javier; Reuther, Gary W; Wright, Kenneth L; Conti, Chiara; Lee, Jennifer Y; Zheng, Xiaozhang; Ng, Pui Yee; Martin, Matthew W; Marshall, C Gary; Koomen, John M; Levine, Ross L; Verma, Amit; Grimes, H Leighton; Sotomayor, Eduardo M; Shao, Zonghong; Epling-Burnette, Pearlie K