Synthesis and structure-activity relationships of 8-(pyrid-3-yl)pyrazolo[1,5-a]-1,3,5-triazines: potent, orally bioavailable corticotropin releasing factor receptor-1 (CRF1) antagonists
8-(吡啶-3-基)吡唑并[1,5-a]-1,3,5-三嗪的合成及构效关系:强效、口服生物可利用的促皮质素释放因子受体-1 (CRF1) 拮抗剂
期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/jm900025h
Paul J Gilligan, Todd Clarke, Liqi He, Snjezana Lelas, Yu-Wen Li, Karen Heman, Lawrence Fitzgerald, Keith Miller, Ge Zhang, Anne Marshall, Carol Krause, John F McElroy, Kathyrn Ward, Kim Zeller, Harvey Wong, Steven Bai, Joanne Saye, Scott Grossman, Robert Zaczek, Stephen P Arneric, Paul Hartig, Davi