日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Tetrameric, active PKM2 inhibits IP3 receptors, potentially requiring GRP75 as an additional interaction partner

四聚体活性 PKM2 抑制 IP3 受体,可能需要 GRP75 作为额外的相互作用伙伴

Fernanda O Lemos, Ian de Ridder, Larry Wagner, Martin D Bootman, Geert Bultynck, David I Yule, Jan B Parys

Intracellular BAPTA directly inhibits PFKFB3, thereby impeding mTORC1-driven Mcl-1 translation and killing MCL-1-addicted cancer cells

细胞内BAPTA直接抑制PFKFB3,从而阻碍mTORC1驱动的Mcl-1翻译,并杀死依赖MCL-1的癌细胞。

Flore Sneyers ,Martijn Kerkhofs ,Femke Speelman-Rooms ,Kirsten Welkenhuyzen ,Rita La Rovere ,Ahmed Shemy ,Arnout Voet ,Guy Eelen ,Mieke Dewerchin ,Stephen W G Tait ,Bart Ghesquière ,Martin D Bootman ,Geert Bultynck

The Complex Effects of PKM2 and PKM2:IP3R Disruption on Intracellular Ca2+ Handling and Cellular Functions

PKM2 和 PKM2:IP3R 功能紊乱对细胞内 Ca2+ 处理和细胞功能的复杂影响

Fernanda O Lemos ,Ian de Ridder ,Martin D Bootman ,Geert Bultynck ,Jan B Parys

Off-target inhibition of NGLY1 by the polycaspase inhibitor Z-VAD-fmk induces cellular autophagy

多聚胱天蛋白酶抑制剂 Z-VAD-fmk 对 NGLY1 的脱靶抑制会诱导细胞自噬

Sarah H Needs, Martin D Bootman, Jeff E Grotzke, Holger B Kramer, Sarah A Allman

A non-canonical role for pyruvate kinase M2 as a functional modulator of Ca2+ signalling through IP3 receptors

丙酮酸激酶 M2 作为通过 IP3 受体传导 Ca2+ 信号的功能调节剂的非典型作用

Andrew R Lavik, Karen S McColl, Fernanda O Lemos, Martijn Kerkhofs, Fei Zhong, Michael Harr, Daniela Schlatzer, Kozo Hamada, Katsuhiko Mikoshiba, Francesco Crea, Geert Bultynck, Martin D Bootman, Jan B Parys, Clark W Distelhorst

Constitutive IP3 signaling underlies the sensitivity of B-cell cancers to the Bcl-2/IP3 receptor disruptor BIRD-2

组成性 IP3 信号是 B 细胞癌症对 Bcl-2/IP3 受体干扰物 BIRD-2 敏感性的基础

Mart Bittremieux, Rita M La Rovere, Haidar Akl, Claudio Martines, Kirsten Welkenhuyzen, Kathia Dubron, Myriam Baes, Ann Janssens, Peter Vandenberghe, Luca Laurenti, Katja Rietdorf, Giampaolo Morciano, Paolo Pinton, Katsuhiko Mikoshiba, Martin D Bootman, Dimitar G Efremov, Humbert De Smedt, Jan B Par

Examining Cardiomyocyte Dysfunction Using Acute Chemical Induction of an Ageing Phenotype

使用急性化学诱导衰老表型检查心肌细胞功能障碍

Said Masoud, Fraser McDonald, Dirk Bister, Claire Kotecki, Martin D Bootman, Katja Rietdorf

Contractile responses to endothelin-1 are regulated by PKC phosphorylation of cardiac myosin binding protein-C in rat ventricular myocytes

大鼠心室肌细胞对内皮素-1 的收缩反应受 PKC 对心肌肌球蛋白结合蛋白-C 的磷酸化调控

Ioannis Smyrnias, Normann Goodwin, Dagmar Wachten, Jonas Skogestad, Jan Magnus Aronsen, Emma L Robinson, Kateryna Demydenko, Anne Segonds-Pichon, David Oxley, Sakthivel Sadayappan, Karin Sipido, Martin D Bootman, H Llewelyn Roderick

Calcium phosphate particles stimulate interleukin-1β release from human vascular smooth muscle cells: A role for spleen tyrosine kinase and exosome release

磷酸钙颗粒刺激人血管平滑肌细胞释放白细胞介素-1β:脾脏酪氨酸激酶和外泌体释放的作用

Yana Dautova, Alexander N Kapustin, Kevin Pappert, Matthias Epple, Hanneke Okkenhaug, Simon J Cook, Catherine M Shanahan, Martin D Bootman, Diane Proudfoot

Oncogenic KRAS suppresses store-operated Ca2+ entry and ICRAC through ERK pathway-dependent remodelling of STIM expression in colorectal cancer cell lines

致癌基因 KRAS 通过 ERK 通路依赖性重塑结直肠癌细胞系中的 STIM 表达来抑制池操纵的 Ca2+ 进入和 ICRAC

Cristina Pierro, Xuexin Zhang, Cynthia Kankeu, Mohamed Trebak, Martin D Bootman, H Llewelyn Roderick