Discovery of the First Orally Available, Selective K(Na)1.1 Inhibitor: In Vitro and In Vivo Activity of an Oxadiazole Series
首个口服选择性K(Na)1.1抑制剂的发现:恶二唑系列化合物的体外和体内活性
期刊:ACS Medicinal Chemistry Letters
影响因子:4
doi:10.1021/acsmedchemlett.0c00675
Griffin, Andrew M; Kahlig, Kristopher M; Hatch, Robert John; Hughes, Zoë A; Chapman, Mark L; Antonio, Brett; Marron, Brian E; Wittmann, Marion; Martinez-Botella, Gabriel