日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Enhanced anticancer effect of thymidylate synthase dimer disrupters by promoting intracellular accumulation.

胸苷酸合成酶二聚体破坏剂通过促进细胞内积累增强抗癌作用

Marverti Gaetano, Moschella Maria Gaetana, Belardo Alice, Lamesta Michele, Mercanile Giada, Tagliazucchi Lorenzo, Aiello Daniele, Venturelli Alberto, Illuminati Davide, Guerrini Remo, Losi Lorena, Ponterini Glauco, Costi Maria Paola, D'Arca Domenico

Targeting the Interplay of Independent Cellular Pathways and Immunity: A Challenge in Cancer Immunotherapy

靶向独立细胞通路与免疫的相互作用:癌症免疫治疗面临的挑战

Lauriola, Angela; Davalli, Pierpaola; Marverti, Gaetano; Santi, Spartaco; Caporali, Andrea; D'Arca, Domenico

Dabrafenib-Panobinostat Salt: Improving the Dissolution Rate and Inhibition of BRAF Melanoma Cells

达拉非尼-帕诺比司他盐:提高溶解速率并抑制BRAF黑色素瘤细胞

Rai, Sunil K; Marverti, Gaetano; Gunnam, Anilkumar; Allu, Suryanarayana; Nangia, Ashwini K

Serum Mass Spectrometry Proteomics and Protein Set Identification in Response to FOLFOX-4 in Drug-Resistant Ovarian Carcinoma

耐药卵巢癌患者对 FOLFOX-4 治疗的反应性血清质谱蛋白质组学和蛋白质组鉴定

Domenico D'Arca, Leda Severi, Stefania Ferrari, Luca Dozza, Gaetano Marverti, Fulvio Magni, Clizia Chinello, Lisa Pagani, Lorenzo Tagliazucchi, Marco Villani, Gianluca d'Addese, Isabella Piga, Vincenza Conteduca, Lorena Rossi, Giorgia Gurioli, Ugo De Giorgi, Lorena Losi, Maria Paola Costi

Identification of a Quinone Derivative as a YAP/TEAD Activity Modulator from a Repurposing Library

从化合物重定位库中鉴定出一种醌衍生物作为YAP/TEAD活性调节剂。

Lauriola, Angela; Uliassi, Elisa; Santucci, Matteo; Bolognesi, Maria Laura; Mor, Marco; Scalvini, Laura; Elisi, Gian Marco; Gozzi, Gaia; Tagliazucchi, Lorenzo; Marverti, Gaetano; Ferrari, Stefania; Losi, Lorena; D'Arca, Domenico; Costi, Maria Paola

Telomere Dysfunction Is Associated with Altered DNA Organization in Trichoplein/Tchp/Mitostatin (TpMs) Depleted Cells

端粒功能障碍与 Trichoplein/Tchp/Mitostatin (TpMs) 耗竭细胞中的 DNA 组织改变有关

Angela Lauriola, Pierpaola Davalli, Gaetano Marverti, Andrea Caporali, Sabine Mai, Domenico D'Arca

Folic Acid-Peptide Conjugates Combine Selective Cancer Cell Internalization with Thymidylate Synthase Dimer Interface Targeting

叶酸-肽结合物将选择性癌细胞内化与胸苷酸合酶二聚体界面靶向相结合

Gaetano Marverti, Chiara Marraccini, Andrea Martello, Domenico D'Arca, Salvatore Pacifico, Remo Guerrini, Francesca Spyrakis, Gaia Gozzi, Angela Lauriola, Matteo Santucci, Giuseppe Cannazza, Lorenzo Tagliazucchi, Addolorata Stefania Cazzato, Lorena Losi, Stefania Ferrari, Glauco Ponterini, Maria P C

Structural Bases for the Synergistic Inhibition of Human Thymidylate Synthase and Ovarian Cancer Cell Growth by Drug Combinations.

药物组合协同抑制人胸苷酸合成酶和卵巢癌细胞生长的结构基础

Pozzi Cecilia, Santucci Matteo, Marverti Gaetano, D'Arca Domenico, Tagliazucchi Lorenzo, Ferrari Stefania, Gozzi Gaia, Losi Lorena, Tassone Giusy, Mangani Stefano, Ponterini Glauco, Costi Maria Paola

A Peptidic Thymidylate-Synthase Inhibitor Loaded on Pegylated Liposomes Enhances the Antitumour Effect of Chemotherapy Drugs in Human Ovarian Cancer Cells

载于聚乙二醇化脂质体的肽类胸苷酸合酶抑制剂增强化疗药物对人类卵巢癌细胞的抗肿瘤作用

Gaetano Marverti, Gaia Gozzi, Eleonora Maretti, Angela Lauriola, Leda Severi, Francesca Sacchetti, Lorena Losi, Salvatore Pacifico, Stefania Ferrari, Glauco Ponterini, Eliana Leo, Maria Paola Costi, Domenico D'Arca

Depletion of Trichoplein (TpMs) Causes Chromosome Mis-Segregation, DNA Damage and Chromosome Instability in Cancer Cells

Trichoplein (TpMs) 的消耗会导致癌细胞中的染色体错误分离、DNA 损伤和染色体不稳定

Angela Lauriola, Andrea Martello, Sebastian Fantini, Gaetano Marverti, Tommaso Zanocco-Marani, Pierpaola Davalli, Daniele Guardavaccaro, Sabine Mai, Andrea Caporali, Domenico D'Arca