Discovery of trans-4-[1-[[2,5-Dichloro-4-(1-methyl-3-indolylcarboxamido)phenyl]acetyl]-(4S)-methoxy-(2S)-pyrrolidinylmethoxy]cyclohexanecarboxylic acid: an orally active, selective very late antigen-4 antagonist
发现反式-4-[1-[[2,5-二氯-4-(1-甲基-3-吲哚基甲酰胺基)苯基]乙酰基]-(4S)-甲氧基-(2S)-吡咯烷基甲氧基]环己烷羧酸:一种口服活性、选择性极晚期抗原-4 拮抗剂
期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/jm901154c
Fumihito Muro, Shin Iimura, Yuuichi Sugimoto, Yoshiyuki Yoneda, Jun Chiba, Toshiyuki Watanabe, Masaki Setoguchi, Yutaka Iigou, Keiko Matsumoto, Atsushi Satoh, Gensuke Takayama, Tomoe Taira, Mika Yokoyama, Tohru Takashi, Atsushi Nakayama, Nobuo Machinaga