日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

The Poly (ADP-ribose) polymerase inhibitor olaparib and pan-ErbB inhibitor neratinib are highly synergistic in HER2 overexpressing epithelial ovarian carcinoma in vitro and in vivo

聚(ADP-核糖)聚合酶抑制剂奥拉帕尼和泛 ErbB 抑制剂来那替尼在体外和体内对 HER2 过度表达的上皮性卵巢癌具有高度协同作用

Chanhee Han, Blair McNamara, Stefania Bellone, Justin Harold, Paola Manara, Tobias Max Philipp Hartwich, Levent Mutlu, Yang Yang-Hartwich, Margherita Zipponi, Cem Demirkiran, Miguel Skyler Z Verzosa, Gary Altwerger, Elena Ratner, Gloria S Huang, Mitchell Clark, Vaagn Andikyan, Masoud Azodi, Peter R

Ovarian and uterine carcinosarcomas are sensitive in vitro and in vivo to elimusertib, a novel ataxia-telangiectasia and Rad3-related (ATR) kinase inhibitor

卵巢癌和子宫癌肉瘤在体内和体外均对 elimusertib 敏感,后者是一种新型共济失调毛细血管扩张症和 Rad3 相关 (ATR) 激酶抑制剂

Diego D Manavella, Blair McNamara, Justin Harold, Stefania Bellone, Tobias Max Philipp Hartwich, Yang Yang-Hartwich, Levent Mutlu, Margherita Zipponi, Cem Demirkiran, Miguel Skyler Verzosa, Gary Altwerger, Elena Ratner, Gloria S Huang, Mitchell Clark, Vaagn Andikyan, Masoud Azodi, Peter E Schwartz, 

Derangements in HUWE1/c-MYC pathway confer sensitivity to the BET bromodomain inhibitor GS-626510 in uterine cervical carcinoma

HUWE1/c-MYC 通路紊乱导致宫颈癌对 BET 溴结构域抑制剂 GS-626510 敏感

Elena Bonazzoli, Stefania Bellone, Luca Zammataro, Barbara Gnutti, Adele Guglielmi, Silvia Pelligra, Nupur Nagarkatti, Paola Manara, Joan Tymon-Rosario, Burak Zeybek, Gary Altwerger, Gulden Menderes, Chanhee Han, Elena Ratner, Dan-Arin Silasi, Gloria S Huang, Vaagn Andikyan, Masoud Azodi, Peter E Sc

Cervical carcinomas that overexpress human trophoblast cell-surface marker (Trop-2) are highly sensitive to the antibody-drug conjugate sacituzumab govitecan

过度表达人类滋养层细胞表面标志物 (Trop-2) 的宫颈癌对抗体-药物偶联物 sacituzumab govitecan 高度敏感

Burak Zeybek, Aranzazu Manzano, Anna Bianchi, Elena Bonazzoli, Stefania Bellone, Natalia Buza, Pei Hui, Salvatore Lopez, Emanuele Perrone, Paola Manara, Luca Zammataro, Gary Altwerger, Chanhee Han, Joan Tymon-Rosario, Gulden Menderes, Elena Ratner, Dan-Arin Silasi, Gloria S Huang, Masoud Azodi, Pete

PARP-1 activity (PAR) determines the sensitivity of cervical cancer to olaparib

PARP-1 活性 (PAR) 决定宫颈癌对奥拉帕尼的敏感性

Anna Bianchi, Salvatore Lopez, Gary Altwerger, Stefania Bellone, Elena Bonazzoli, Luca Zammataro, Aranzazu Manzano, Paola Manara, Emanuele Perrone, Burak Zeybek, Chanhee Han, Gulden Menderes, Elena Ratner, Dan-Arin Silasi, Gloria S Huang, Masoud Azodi, Justin Y Newberg, Dean C Pavlick, Julia Elvin, 

PIK3CA oncogenic mutations represent a major mechanism of resistance to trastuzumab in HER2/neu overexpressing uterine serous carcinomas

PIK3CA 致癌突变是 HER2/neu 过度表达的子宫浆液性癌对曲妥珠单抗产生耐药性的主要机制

Jonathan D Black, Salvatore Lopez, Emiliano Cocco, Stefania Bellone, Gary Altwerger, Carlton L Schwab, Diana P English, Elena Bonazzoli, Federica Predolini, Francesca Ferrari, Elena Ratner, Dan-Arin Silasi, Masoud Azodi, Peter E Schwartz, Alessandro D Santin

Dual HER2/PIK3CA Targeting Overcomes Single-Agent Acquired Resistance in HER2-Amplified Uterine Serous Carcinoma Cell Lines In Vitro and In Vivo

HER2/PIK3CA 双靶向治疗在体内和体外克服了 HER2 扩增子宫浆液性癌细胞系中单药获得性耐药性

Salvatore Lopez, Emiliano Cocco, Jonathan Black, Stefania Bellone, Elena Bonazzoli, Federica Predolini, Francesca Ferrari, Carlton L Schwab, Diana P English, Elena Ratner, Dan-Arin Silasi, Masoud Azodi, Peter E Schwartz, Corrado Terranova, Roberto Angioli, Alessandro D Santin

Polymerase ε (POLE) ultra-mutated tumors induce robust tumor-specific CD4+ T cell responses in endometrial cancer patients

聚合酶 ε (POLE) 超突变肿瘤在子宫内膜癌患者中诱导强烈的肿瘤特异性 CD4+ T 细胞反应

Stefania Bellone, Floriana Centritto, Jonathan Black, Carlton Schwab, Diana English, Emiliano Cocco, Salvatore Lopez, Elena Bonazzoli, Federica Predolini, Francesca Ferrari, Dan-Arin Silasi, Elena Ratner, Masoud Azodi, Peter E Schwartz, Alessandro D Santin

Dacomitinib (PF-00299804), a second-generation irreversible pan-erbB receptor tyrosine kinase inhibitor, demonstrates remarkable activity against HER2-amplified uterine serous endometrial cancer in vitro

达克替尼 (PF-00299804) 是一种第二代不可逆泛 erbB 受体酪氨酸激酶抑制剂,体外对 HER2 扩增的子宫浆液性子宫内膜癌表现出显著的活性

Liancheng Zhu, Salvatore Lopez, Stefania Bellone, Jonathan Black, Emiliano Cocco, Tiffany Zigras, Federica Predolini, Elena Bonazzoli, Beatrice Bussi, Zachary Stuhmer, Carlton L Schwab, Diana P English, Elena Ratner, Dan-Arin Silasi, Masoud Azodi, Peter E Schwartz, Thomas J Rutherford, Alessandro D

Class III β-tubulin overexpression within the tumor microenvironment is a prognostic biomarker for poor overall survival in ovarian cancer patients treated with neoadjuvant carboplatin/paclitaxel

肿瘤微环境中 III 类 β-微管蛋白过度表达是接受新辅助卡铂/紫杉醇治疗的卵巢癌患者总体生存率较差的预后生物标志物

Dana M Roque, Natalia Buza, Michelle Glasgow, Stefania Bellone, Ileana Bortolomai, Sara Gasparrini, Emiliano Cocco, Elena Ratner, Dan-Arin Silasi, Masoud Azodi, Thomas J Rutherford, Peter E Schwartz, Alessandro D Santin