日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Modulators of Diacylglycerol Kinase Activity: A Review of Advances and Challenges

二酰甘油激酶活性调节剂:进展与挑战综述

Racca, Luisa; Baldanzi, Gianluca; Massarotti, Alberto

Development of PROTACs Targeting the Moonlighting Enzyme Nicotinamide Phosphoribosyltransferase (NAMPT) for Breast Cancer Therapy

开发靶向多功能酶烟酰胺磷酸核糖转移酶 (NAMPT) 的 PROTAC 用于乳腺癌治疗

Galli, Ubaldina; Moro, Marianna; Balestrero, Federica Carolina; Colombo, Giorgia; Koten, Marco; Roncaglio, Benedetta; Genazzani, Armando A; Aprile, Silvio; Massarotti, Alberto; Orsomando, Giuseppe; Pirali, Tracey; Grolla, Ambra A

Structure-Guided Optimization and Biological Validation of 1,3,4-Thiadiazole-Based SIRT2 Inhibitors Reinforcing Channel Entrance Interactions.

基于结构的 1,3,4-噻二唑 SIRT2 抑制剂的优化和生物学验证,增强了通道入口相互作用。

Aksel Ahmet Bugra, Ozgencil Fikriye, Bakar-Ates Filiz, Gunindi Habibe Beyza, Massarotti Alberto, Ozkan Erva, Kaya Selen Gozde, Gozelle Mahmut, Ozkan Yesim, Eren Gokcen

Acute Myeloid Leukemia: A Key Role of DGKα and DGKζ in Cell Viability

急性髓系白血病:DGKα和DGKζ在细胞存活中的关键作用

Gorla, Elisa; Cartella, Marco Cristiano; Borghetti, Edoardo; Lovati, Ginevra; Racca, Luisa; Gravina, Teresa; Biazzo, Giorgio; Bonello, Gabriele; Malacarne, Valeria; De Giorgis, Veronica; Corà, Davide; Manfredi, Marcello; Massarotti, Alberto; Graziani, Andrea; Baldanzi, Gianluca

Arzanol Inhibits Human Dihydroorotate Dehydrogenase and Shows Antiviral Activity

Arzanol抑制人二氢乳清酸脱氢酶并显示出抗病毒活性

Alberti, Marta; Tamburello, Martina; Salamone, Stefano; Gallinella, Giorgio; Sanna, Cinzia; Appendino, Giovanni Battista; Lolli, Marco L; Massarotti, Alberto; Pollastro, Federica; Miggiano, Riccardo

A nonnatural peptide targeting the A-kinase anchoring function of PI3Kγ for therapeutic cAMP modulation in pulmonary cells

一种靶向PI3Kγ的A激酶锚定功能的非天然肽,用于肺细胞中cAMP的治疗性调节。

Della Sala, Angela; Tasca, Laura; Butnarasu, Cosmin; Sala, Valentina; Prono, Giulia; Murabito, Alessandra; Garbero, Olga Valentina; Millo, Enrico; Terranova, Leonardo; Blasi, Francesco; Gramegna, Andrea; Aliberti, Stefano; Massarotti, Alberto; Visentin, Sonja; Hirsch, Emilio; Ghigo, Alessandra

Identification of a Compound Inhibiting Both the Enzymatic and Nonenzymatic Functions of Indoleamine 2,3-Dioxygenase 1.

鉴定一种抑制吲哚胺 2,3-双加氧酶 1 的酶促和非酶促功能的化合物

Panfili Eleonora, Rezzi Sarah Jane, Adamo Annalisa, Mazzoletti Daniele, Massarotti Alberto, Miggiano Riccardo, Fallarini Silvia, Ambrosino Sara, Coletti Alice, Molinaro Pasquale, Milella Michele, Paiella Salvatore, Macchiarulo Antonio, Ugel Stefano, Pirali Tracey, Pallotta Maria Teresa

What's in a Name? Drug Nomenclature and Medicinal Chemistry Trends using INN Publications

名称的意义何在?基于国际非专利名称(INN)出版物的药物命名和药物化学趋势

Serafini, Marta; Cargnin, Sarah; Massarotti, Alberto; Tron, Gian Cesare; Pirali, Tracey; Genazzani, Armando A

The SNAP-tag technology revised: an effective chemo-enzymatic approach by using a universal azide-based substrate

SNAP标签技术的改进:一种利用通用叠氮化物底物的有效化学酶法

Merlo, Rosa; Caprioglio, Diego; Cillo, Michele; Valenti, Anna; Mattossovich, Rosanna; Morrone, Castrese; Massarotti, Alberto; Rossi, Franca; Miggiano, Riccardo; Leonardi, Antonio; Minassi, Alberto; Perugino, Giuseppe

Essential Medicinal Chemistry of Essential Medicines

基本药物的基本药物化学

Serafini, Marta; Cargnin, Sarah; Massarotti, Alberto; Pirali, Tracey; Genazzani, Armando A