日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Discovery and development of a new oxazolidinone with reduced toxicity for the treatment of tuberculosis

发现和开发一种毒性降低的新型噁唑烷酮类药物用于治疗结核病

Crowley, Brendan M; Boshoff, Helena I; Boving, Aidan; Tan, Vee Y; Zhu, Jianghai; Hoyt, Forrest; Miller, Randy R; Ehrhart, Julie; Boyce, Christopher W; Young, Katherine; Nantermet, Philippe G; Su, Jing; Yang, Lihu; Painter, Ronald E; Corcoran, Emily B; Hoar, Jason L; Oh, Sangmi; Holtzman, David L; Levi, Micha; Anderson, Aparna; Otieno, Monicah A; Zimmerman, Matthew; Kaya, Firat; Massoudi, Lisa M; Ramey, Michelle E; Bauman, Allison A; Lenaerts, Anne J; Roberston, Gregory T; Dartois, Véronique; Wells, Charles D; Barry, Clifton E 3rd; Olsen, David B

Physiologic recovery of Mycobacterium tuberculosis from drug injury: A molecular study of post antibiotic effect in vitro and in vivo

结核分枝杆菌药物损伤后的生理恢复:体外和体内抗生素后效应的分子研究

Hendrix, Jo; Al Mubarak, Reem; Reichlen, Matthew J; Tabor, Samuel T; Bateman, Adeline; Massoudi, Lisa M; Rossmassler, Karen; Kaya, Firat; Zimmerman, Matthew D; Nielsen, Holly; Wynn, Elizabeth A; Voskuil, Martin I; Robertson, Gregory T; Moore, Camille M; Walter, Nicholas D

SuFEx-based antitubercular compound irreversibly inhibits Pks13

基于 SuFEx 的抗结核化合物不可逆地抑制 Pks13

Krieger, Inna V; Sukheja, Paridhi; Yang, Baiyuan; Tang, Su; Selle, Daniel; Woods, Ashley; Engelhart, Curtis; Kumar, Pradeep; Harbut, Michael B; Liu, Dongdong; Tsuda, Brendan; Qin, Bo; Bare, Grant A L; Li, Gencheng; Chi, Victor; Gambacurta, Julian; Hvizdos, Janine; Reagan, Matthew; Jones, Isabelle L; Massoudi, Lisa M; Woolhiser, Lisa K; Cascioferro, Alessandro; Kundrick, Erica; Singh, Parul; Reiley, William; Ioerger, Thomas R; Kandula, Dilipkumar Reddy; McCabe, Jacob W; Guo, Taijie; Alland, David; Boshoff, Helena I; Schnappinger, Dirk; Robertson, Gregory T; Mdluli, Khisi; Lee, Kyoung-Jin; Dong, Jiajia; Li, Shuangwei; Schultz, Peter G; Joseph, Sean B; Love, Melissa S; Sharpless, K Barry; Petrassi, H Michael; Chatterjee, Arnab K; Sacchettini, James C; McNamara, Case W

Emergence of antibiotic-specific Mycobacterium tuberculosis phenotypes during prolonged treatment of mice

小鼠长期治疗过程中出现抗生素特异性结核分枝杆菌表型

Wynn, Elizabeth A; Dide-Agossou, Christian; Al Mubarak, Reem; Rossmassler, Karen; Ektnitphong, Victoria; Bauman, Allison A; Massoudi, Lisa M; Voskuil, Martin I; Robertson, Gregory T; Moore, Camille M; Walter, Nicholas D

Spectinamide MBX-4888A exhibits favorable lesion and tissue distribution and promotes treatment shortening in advanced murine models of tuberculosis

Spectinamide MBX-4888A 在晚期小鼠结核病模型中表现出良好的病灶和组织分布,并能缩短治疗时间。

Bauman, Allison A; Sarathy, Jansy P; Kaya, Firat; Massoudi, Lisa M; Scherman, Michael S; Hastings, Courtney; Liu, Jiuyu; Xie, Min; Brooks, Elizabeth J; Ramey, Michelle E; Jones, Isabelle L; Benedict, Noalani D; Maclaughlin, Madelyn R; Miller-Dawson, Jake A; Waidyarachchi, Samanthi L; Butler, Michelle M; Bowlin, Terry L; Zimmerman, Matthew D; Lenaerts, Anne J; Meibohm, Bernd; Gonzalez-Juarrero, Mercedes; Lyons, Michael A; Dartois, Veronique; Lee, Richard E; Robertson, Gregory T

Transcriptional adaptation of Mycobacterium tuberculosis that survives prolonged multi-drug treatment in mice

结核分枝杆菌在小鼠体内长期多药治疗后存活的转录适应

Wynn, Elizabeth A; Dide-Agossou, Christian; Reichlen, Matthew; Rossmassler, Karen; Al Mubarak, Reem; Reid, Justin J; Tabor, Samuel T; Born, Sarah E M; Ransom, Monica R; Davidson, Rebecca M; Walton, Kendra N; Benoit, Jeanne B; Hoppers, Amanda; Loy, Dorothy E; Bauman, Allison A; Massoudi, Lisa M; Dolganov, Gregory; Strong, Michael; Nahid, Payam; Voskuil, Martin I; Robertson, Gregory T; Moore, Camille M; Walter, Nicholas D

Drug distribution and efficacy of the DprE1 inhibitor BTZ-043 in the C3HeB/FeJ mouse tuberculosis model.

DprE1抑制剂BTZ-043在C3HeB/FeJ小鼠结核病模型中的药物分布和疗效

Ramey Michelle E, Kaya Firat, Bauman Allison A, Massoudi Lisa M, Sarathy Jansy P, Zimmerman Matthew D, Scott Dashick W L, Job Alyx M, Miller-Dawson Jake A, Podell Brendan K, Lyons Michael A, Dartois Véronique, Lenaerts Anne J, Robertson Gregory T

Transcriptional adaptation of drug-tolerant Mycobacterium tuberculosis in mice

小鼠体内耐药结核分枝杆菌的转录适应

Wynn, Elizabeth A; Dide-Agossou, Christian; Reichlen, Matthew; Rossmassler, Karen; Al Mubarak, Reem; Reid, Justin J; Tabor, Samuel T; Born, Sarah E M; Ransom, Monica R; Davidson, Rebecca M; Walton, Kendra N; Benoit, Jeanne B; Hoppers, Amanda; Bauman, Allison A; Massoudi, Lisa M; Dolganov, Gregory; Nahid, Payam; Voskuil, Martin I; Robertson, Gregory T; Moore, Camille M; Walter, Nicholas D

Optimization of TAM16, a Benzofuran That Inhibits the Thioesterase Activity of Pks13; Evaluation toward a Preclinical Candidate for a Novel Antituberculosis Clinical Target

优化TAM16(一种抑制Pks13硫酯酶活性的苯并呋喃类化合物);评估其作为新型抗结核临床靶点的临床前候选药物

Wilson, Caroline; Ray, Peter; Zuccotto, Fabio; Hernandez, Jorge; Aggarwal, Anup; Mackenzie, Claire; Caldwell, Nicola; Taylor, Malcolm; Huggett, Margaret; Mathieson, Michael; Murugesan, Dinakaran; Smith, Alasdair; Davis, Susan; Cocco, Mattia; Parai, Maloy K; Acharya, Arjun; Tamaki, Fabio; Scullion, Paul; Epemolu, Ola; Riley, Jennifer; Stojanovski, Laste; Lopez-Román, Eva Maria; Torres-Gómez, Pedro Alfonso; Toledo, Ana Maria; Guijarro-Lopez, Laura; Camino, Isabel; Engelhart, Curtis A; Schnappinger, Dirk; Massoudi, Lisa M; Lenaerts, Anne; Robertson, Gregory T; Walpole, Chris; Matthews, David; Floyd, David; Sacchettini, James C; Read, Kevin D; Encinas, Lourdes; Bates, Robert H; Green, Simon R; Wyatt, Paul G

Spiropyrimidinetriones: a Class of DNA Gyrase Inhibitors with Activity against Mycobacterium tuberculosis and without Cross-Resistance to Fluoroquinolones

螺嘧啶三酮类:一类对结核分枝杆菌具有活性且与氟喹诺酮类药物无交叉耐药性的DNA促旋酶抑制剂

Basarab, Gregory S; Ghorpade, Sandeep; Gibhard, Liezl; Mueller, Rudolf; Njoroge, Mathew; Peton, Nashied; Govender, Preshendren; Massoudi, Lisa M; Robertson, Gregory Thomas; Lenaerts, Anne J; Boshoff, Helena Ingrid; Joerss, Douglas; Parish, Tanya; Durand-Reville, Thomas F; Perros, Manos; Singh, Vinayak; Chibale, Kelly