日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Early Development of Ocadusertib, a Selective Receptor-Interacting Serine/Threonine-Protein Kinase 1 Inhibitor

Ocadusertib(一种选择性受体相互作用丝氨酸/苏氨酸蛋白激酶 1 抑制剂)的早期研发

Shaw, Simon J; Taylor, Vanessa C; Sims, Jonathan T; Ho, Stephen; Lamagna, Chrystelle; Yan, Lucy; Reising, Nicholas C; Chow, Andrew; Hanson, Eric P; Vendel, Andrew C; Dairaghi, Daniel J; Masuda, Esteban S

Randomized Trial on the Effect of an Oral Spleen Tyrosine Kinase Inhibitor in the Treatment of IgA Nephropathy

口服脾酪氨酸激酶抑制剂治疗IgA肾病疗效的随机试验

Tam, Frederick W K; Tumlin, James; Barratt, Jonathan; Rovin, Brad H; Roberts, Ian S D; Roufosse, Candice; Cook, H Terence; Bhangal, Gurjeet; Brown, Alison L; Busch, Martin; Dudhiya, Fayaz; Duliege, Anne-Marie; Fraser, Donald J; Gale, Daniel P; Huang, Chiu-Ching; Lai, Ping-Chin; Lee, Meng; Masuda, Esteban S; McAdoo, Stephen P; Rosenkranz, Alexander R; Sommerer, Claudia; Sunder-Plassmann, Gere; Szeto, Cheuk-Chun; Tang, Sydney C W; Williamson, Don E; Willcocks, Lisa; Vielhauer, Volker; Kim, Min Jeong; Todd, Leslie; Zayed, Hany; Tong-Starksen, Sandra; Lafayette, Richard

Spleen tyrosine kinase inhibition is an effective treatment for established vasculitis in a pre-clinical model

在临床前模型中,脾酪氨酸激酶抑制剂是治疗已确诊血管炎的有效方法。

McAdoo, Stephen P; Prendecki, Maria; Tanna, Anisha; Bhatt, Tejal; Bhangal, Gurjeet; McDaid, John; Masuda, Esteban S; Cook, H Terence; Tam, Frederick W K; Pusey, Charles D

Inhibition of spleen tyrosine kinase prevents mast cell activation and airway hyperresponsiveness

抑制脾酪氨酸激酶可阻止肥大细胞活化和气道高反应性

Matsubara, Shigeki; Li, Guiming; Takeda, Katsuyuki; Loader, Joan E; Pine, Polly; Masuda, Esteban S; Miyahara, Nobuaki; Miyahara, Satoko; Lucas, Joseph J; Dakhama, Azzeddine; Gelfand, Erwin W

Syk activation in dendritic cells is essential for airway hyperresponsiveness and inflammation

树突状细胞中Syk的激活对于气道高反应性和炎症至关重要。

Matsubara, Shigeki; Koya, Toshiyuki; Takeda, Katsuyuki; Joetham, Anthony; Miyahara, Nobuaki; Pine, Polly; Masuda, Esteban S; Swasey, Christina H; Gelfand, Erwin W

Systematic identification of regulatory proteins critical for T-cell activation.

系统性鉴定对T细胞活化至关重要的调控蛋白

Chu Peter, Pardo Jorge, Zhao Haoran, Li Connie C, Pali Erlina, Shen Mary M, Qu Kunbin, Yu Simon X, Huang Betty Cb, Yu Peiwen, Masuda Esteban S, Molineaux Susan M, Kolbinger Frank, Aversa Gregorio, de Vries Jan, Payan Donald G, Liao X Charlene