日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Molecular basis of CXC chemokine receptor 3 ligand multispecificity

CXC趋化因子受体3配体多特异性的分子基础

Bouyssou, Alexandre; Sun, Dawei; Zhou, Tricia; Smith, Shannon; Ho, Hoangdung; Johnson, Matthew; Azumaya, Caleigh; Noreng, Sigrid; Liu, Peter; Ti, Shu; Joshi, Prajakta; Tam, Christine; Yang, Ying; Janezic, Eric; Comps-Agrar, Laëtitia; Masureel, Matthieu

A Machine Learning-Enabled Venom Peptide Platform for Rapid Drug Discovery.

基于机器学习的毒液肽平台,用于快速药物发现。

Cai Fei, Zhou Lijuan, Delgado Bryce, Chang Wenping, Tom Jeffrey, Hernandez Evelyn, Joshi Prajakta, Song Aimin, Masureel Matthieu, Maun Henry R, Chang Andrew, Zhang Yingnan

Engineered IL-18 variants with half-life extension and improved stability for cancer immunotherapy.

经基因工程改造的IL-18变体,具有延长半衰期和提高稳定性,可用于癌症免疫治疗

Bainbridge Travis W, Wang Lifen, Moskalenko Marina, Herrera Robert, Paluch Maciej T, Sun Dawei, Tasneem Kazi, Saini Harpinder, Sadek Manal, Kwong Mandy, Kim Yoon Min, Bhatt Jay M, Tam Christine, Chan Pamela Pui Fung, Ovacik Ayse Meric, Masureel Matthieu, Zhao Yue, Sockolosky Jonathan T, Qu Yan, West Nathaniel R, Bulutoglu Beyza

Membrane phosphoinositides allosterically tune β-arrestin dynamics to facilitate GPCR core engagement

膜磷脂酰肌醇通过变构调节β-arrestin的动力学,从而促进GPCR核心的结合。

Janetzko, John; Deutsch, Jonathan; Shi, Yuqi; Siepe, Dirk H; Masureel, Matthieu; Liu, Weijing; Viner, Rosa; Inoue, Asuka; Chu, Steven; Kobilka, Brian K; Shivnaraine, Rabindra V

Structure of the neurotensin receptor 1 in complex with β-arrestin 1.

神经降压素受体 1 与 β-arrestin 1 复合物的结构

Huang Weijiao, Masureel Matthieu, Qu Qianhui, Janetzko John, Inoue Asuka, Kato Hideaki E, Robertson Michael J, Nguyen Khanh C, Glenn Jeffrey S, Skiniotis Georgios, Kobilka Brian K

An embedded lipid in the multidrug transporter LmrP suggests a mechanism for polyspecificity

多药转运蛋白LmrP中嵌入的脂质提示了一种多特异性机制

Debruycker, Vincent; Hutchin, Andrew; Masureel, Matthieu; Ficici, Emel; Martens, Chloé; Legrand, Pierre; Stein, Richard A; Mchaourab, Hassane S; Faraldo-Gómez, José D; Remaut, Han; Govaerts, Cédric

Structure and dynamics of GPCR signaling complexes

GPCR信号复合物的结构和动力学

Hilger, Daniel; Masureel, Matthieu; Kobilka, Brian K

Allosteric regulation of G protein-coupled receptor activity by phospholipids

磷脂对G蛋白偶联受体活性的变构调节

Dawaliby, Rosie; Trubbia, Cataldo; Delporte, Cédric; Masureel, Matthieu; Van Antwerpen, Pierre; Kobilka, Brian K; Govaerts, Cédric

Protonation drives the conformational switch in the multidrug transporter LmrP

质子化驱动多药转运蛋白LmrP的构象转变

Masureel, Matthieu; Martens, Chloé; Stein, Richard A; Mishra, Smriti; Ruysschaert, Jean-Marie; Mchaourab, Hassane S; Govaerts, Cédric