日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Native Taylor/Non-Taylor Dispersion-Mass Spectrometry (TNT-MS) Allows Rapid Protein Desalting and Multiplexed, Label-Free Ligand Screening

原生泰勒/非泰勒色散质谱(TNT-MS)可实现快速蛋白质脱盐和多重无标记配体筛选

Eisert, Jonathan; Maciel, Edvaldo Vasconcelos Soares; Dederer, Verena; Berwanger, Aylin; Bailey, Henry J; Đikić, Ivan; Knapp, Stefan; Empting, Martin; Mathea, Sebastian; Jensen, Henrik; Lermyte, Frederik

Type II kinase inhibitors that target Parkinson's disease-associated LRRK2

靶向帕金森病相关LRRK2的II型激酶抑制剂

Nicolai D Raig ,Katherine J Surridge ,Marta Sanz-Murillo ,Verena Dederer ,Andreas Krämer ,Martin P Schwalm ,Nicholas M Lattal ,Lewis Elson ,Deep Chatterjee ,Sebastian Mathea ,Thomas Hanke ,Andres E Leschziner ,Samara L Reck-Peterson ,Stefan Knapp

Correction: LRRK2 dynamics analysis identifies allosteric control of the crosstalk between its catalytic domains

更正:LRRK2动力学分析揭示了其催化结构域间串扰的变构调控

Weng, Jui-Hung; Aoto, Phillip C; Lorenz, Robin; Wu, Jian; Schmidt, Sven H; Manschwetus, Jascha T; Kaila-Sharma, Pallavi; Silletti, Steve; Torres-Paris, Constanza; Mathea, Sebastian; Chatterjee, Deep; Knapp, Stefan; Herberg, Friedrich W; Taylor, Susan S

Covalent Targeting Leads to the Development of a LIMK1 Isoform-Selective Inhibitor

共价靶向导致LIMK1亚型选择性抑制剂的开发

Sebastian Mandel ,Thomas Hanke ,Niall Prendiville ,María Baena-Nuevo ,Lena Marie Berger ,Frederic Farges ,Martin Peter Schwalm ,Benedict-Tilman Berger ,Andreas Kraemer ,Lewis Elson ,Hayuningbudi Saraswati ,Kamal R Abdul Azeez ,Verena Dederer ,Sebastian Mathea ,Ana Corrionero ,Patricia Alfonso ,Sabrina Keller ,Matthias Gstaiger ,Daniela S Krause ,Susanne Müller ,Sandra Röhm ,Stefan Knapp

Aligning With the Goals of the Planetary Health Concept Regarding Ecological Sustainability and Digital Health: Scoping Review

与地球健康理念在生态可持续性和数字健康方面的目标相一致:范围界定综述

Berger, Mathea; Ehlers, Jan Peter; Nitsche, Julia

Development of pyrazolo[1,5-a]pyrimidine based macrocyclic kinase inhibitors targeting AAK1.

开发以吡唑并[1,5-a]嘧啶为基础的大环激酶抑制剂,靶向AAK1。

Mensing Theresa E, Kurz Christian G, Amrhein Jennifer A, Ehret Theresa A L, Preuss Franziska, Mathea Sebastian, Karim Marwah, Tran Do Hoang Nhu, Kadlecova Zuzana, Tolvanen Tuomas A, Martinez-Molina Daniel, Müller Susanne, Einav Shirit, Knapp Stefan, Hanke Thomas

Evaluating Machine Learning Models for Molecular Property Prediction: Performance and Robustness on Out-of-Distribution Data

评估用于分子性质预测的机器学习模型:在分布外数据上的性能和鲁棒性

Fooladi, Hosein; Vu, Thi Ngoc Lan; Mathea, Miriam; Kirchmair, Johannes

Selectivity profiles and substrate recognition of Rab-phosphorylating kinases.

Rab磷酸化激酶的选择性特征和底物识别。

Chatterjee Deep, Dederer Verena, Nguyen Landon Vu, Wendel Marcel, Abdul Azeez Kamal R, Mahesula Swetha, Stengel Florian, Reck-Peterson Samara, Mathea Sebastian

Repurposing of the RIPK1-Selective Benzo[1,4]oxazepin-4-one Scaffold for the Development of a Type III LIMK1/2 Inhibitor.

RIPK1 选择性苯并[1,4]氧氮杂环庚酮-4-酮骨架的再利用,用于开发 III 型 LIMK1/2 抑制剂

Mandel Sebastian, Hanke Thomas, Mathea Sebastian, Chatterjee Deep, Saraswati Hayuningbudi, Berger Benedict-Tilman, Schwalm Martin Peter, Yamamoto Satoshi, Tawada Michiko, Takagi Terufumi, Ahmed Mahmood, Röhm Sandra, Corrionero Ana, Alfonso Patricia, Baena Maria, Elson Lewis, Menge Amelie, Krämer Andreas, Pereira Raquel, Müller Susanne, Krause Daniela S, Knapp Stefan

Impact of face masks on empathy and communication in head and neck cancer patients: a case-control study

口罩对头颈癌患者同理心和沟通能力的影响:一项病例对照研究

Hoene, Georg; von Hahn, Nikolaus; Mathea, Tim; Schminke, Boris; Goldstein, Kathi; Leu, Martin; Schliephake, Henning; Wolfer, Susanne