日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Native Taylor/Non-Taylor Dispersion-Mass Spectrometry (TNT-MS) Allows Rapid Protein Desalting and Multiplexed, Label-Free Ligand Screening

原生泰勒/非泰勒色散质谱(TNT-MS)可实现快速蛋白质脱盐和多重无标记配体筛选

Eisert, Jonathan; Maciel, Edvaldo Vasconcelos Soares; Dederer, Verena; Berwanger, Aylin; Bailey, Henry J; Đikić, Ivan; Knapp, Stefan; Empting, Martin; Mathea, Sebastian; Jensen, Henrik; Lermyte, Frederik

Correction: LRRK2 dynamics analysis identifies allosteric control of the crosstalk between its catalytic domains

更正:LRRK2动力学分析揭示了其催化结构域间串扰的变构调控

Weng, Jui-Hung; Aoto, Phillip C; Lorenz, Robin; Wu, Jian; Schmidt, Sven H; Manschwetus, Jascha T; Kaila-Sharma, Pallavi; Silletti, Steve; Torres-Paris, Constanza; Mathea, Sebastian; Chatterjee, Deep; Knapp, Stefan; Herberg, Friedrich W; Taylor, Susan S

Development of pyrazolo[1,5-a]pyrimidine based macrocyclic kinase inhibitors targeting AAK1.

开发以吡唑并[1,5-a]嘧啶为基础的大环激酶抑制剂,靶向AAK1。

Mensing Theresa E, Kurz Christian G, Amrhein Jennifer A, Ehret Theresa A L, Preuss Franziska, Mathea Sebastian, Karim Marwah, Tran Do Hoang Nhu, Kadlecova Zuzana, Tolvanen Tuomas A, Martinez-Molina Daniel, Müller Susanne, Einav Shirit, Knapp Stefan, Hanke Thomas

Selectivity profiles and substrate recognition of Rab-phosphorylating kinases.

Rab磷酸化激酶的选择性特征和底物识别。

Chatterjee Deep, Dederer Verena, Nguyen Landon Vu, Wendel Marcel, Abdul Azeez Kamal R, Mahesula Swetha, Stengel Florian, Reck-Peterson Samara, Mathea Sebastian

Repurposing of the RIPK1-Selective Benzo[1,4]oxazepin-4-one Scaffold for the Development of a Type III LIMK1/2 Inhibitor.

RIPK1 选择性苯并[1,4]氧氮杂环庚酮-4-酮骨架的再利用,用于开发 III 型 LIMK1/2 抑制剂

Mandel Sebastian, Hanke Thomas, Mathea Sebastian, Chatterjee Deep, Saraswati Hayuningbudi, Berger Benedict-Tilman, Schwalm Martin Peter, Yamamoto Satoshi, Tawada Michiko, Takagi Terufumi, Ahmed Mahmood, Röhm Sandra, Corrionero Ana, Alfonso Patricia, Baena Maria, Elson Lewis, Menge Amelie, Krämer Andreas, Pereira Raquel, Müller Susanne, Krause Daniela S, Knapp Stefan

LRRK2 dynamics analysis identifies allosteric control of the crosstalk between its catalytic domains

LRRK2动力学分析揭示了其催化结构域间相互作用的变构调控

Weng, Jui-Hung; Aoto, Phillip C; Lorenz, Robin; Wu, Jian; Schmidt, Sven H; Manschwetus, Jascha T; Kaila-Sharma, Pallavi; Silletti, Steve; Mathea, Sebastian; Chatterjee, Deep; Knapp, Stefan; Herberg, Friedrich W; Taylor, Susan S

Structural Aspects of LIMK Regulation and Pharmacology

LIMK调控和药理学的结构方面

Chatterjee, Deep; Preuss, Franziska; Dederer, Verena; Knapp, Stefan; Mathea, Sebastian

Trypsiligase-Catalyzed Labeling of Proteins on Living Cells

胰蛋白酶连接酶催化活细胞蛋白质标记

Liebscher, Sandra; Mathea, Sebastian; Aumüller, Tobias; Pech, Andreas; Bordusa, Frank

Lessons from LIMK1 enzymology and their impact on inhibitor design.

从 LIMK1 酶学中汲取的经验教训及其对抑制剂设计的影响

Salah Eidarus, Chatterjee Deep, Beltrami Alessandra, Tumber Anthony, Preuss Franziska, Canning Peter, Chaikuad Apirat, Knaus Petra, Knapp Stefan, Bullock Alex N, Mathea Sebastian

Sfp-type 4'-phosphopantetheinyl transferase is indispensable for fungal pathogenicity

SFP型4'-磷酸泛酰巯基转移酶对真菌致病性至关重要

Horbach, Ralf; Graf, Alexander; Weihmann, Fabian; Antelo, Luis; Mathea, Sebastian; Liermann, Johannes C; Opatz, Till; Thines, Eckhard; Aguirre, Jesús; Deising, Holger B