日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Maintenance of p-eIF2α levels by the eIF2B complex is vital for colorectal cancer

eIF2B复合物维持p-eIF2α水平对结直肠癌至关重要。

Ivana Paskov Škapik # ,Chiara Giacomelli # ,Sarah Hahn ,Hanna Deinlein ,Peter Gallant ,Mathias Diebold ,Josep Biayna ,Anne Hendricks ,Leon Olimski ,Christoph Otto ,Carolin Kastner ,Elmar Wolf ,Christina Schülein-Völk ,Katja Maurus ,Andreas Rosenwald ,Nikolai Schleussner ,Rene-Filip Jackstadt ,Nicolas Schlegel ,Christoph-Thomas Germer ,Martin Bushell ,Martin Eilers ,Stefanie Schmidt ,Armin Wiegering

Identification of suitable target/E3 ligase pairs for PROTAC development using a rapamycin-induced proximity assay (RiPA)

使用雷帕霉素诱导的邻近分析 (RiPA) 鉴定适合 PROTAC 开发的靶标/E3 连接酶对

Bikash Adhikari, Katharina Schneider, Mathias Diebold, Christoph Sotriffer, Elmar Wolf

PROTAC-mediated degradation reveals a non-catalytic function of AURORA-A kinase

PROTAC 介导的降解揭示了 AURORA-A 激酶的非催化功能

Bikash Adhikari #, Jelena Bozilovic #, Mathias Diebold, Jessica Denise Schwarz, Julia Hofstetter, Martin Schröder, Marek Wanior, Ashwin Narain, Markus Vogt, Nevenka Dudvarski Stankovic, Apoorva Baluapuri, Lars Schönemann, Lorenz Eing, Pranjali Bhandare, Bernhard Kuster, Andreas Schlosser, Stephanie

Autoinhibition Mechanism of the Ubiquitin-Conjugating Enzyme UBE2S by Autoubiquitination

泛素结合酶 UBE2S 的自身泛素化抑制机制

Anna K L Liess, Alena Kucerova, Kristian Schweimer, Lu Yu, Theodoros I Roumeliotis, Mathias Diebold, Olexandr Dybkov, Christoph Sotriffer, Henning Urlaub, Jyoti S Choudhary, Jörg Mansfeld, Sonja Lorenz