Discovery and optimization of an azetidine chemical series as a free fatty acid receptor 2 (FFA2) antagonist: from hit to clinic
发现和优化氮杂环丁烷系列化合物作为游离脂肪酸受体 2 (FFA2) 拮抗剂:从热门药物到临床
期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/jm5012885
Mathieu Pizzonero, Sonia Dupont, Marielle Babel, Stéphane Beaumont, Natacha Bienvenu, Roland Blanqué, Laëtitia Cherel, Thierry Christophe, Benedetta Crescenzi, Elsa De Lemos, Philippe Delerive, Pierre Deprez, Steve De Vos, Fatoumata Djata, Stephen Fletcher, Sabrina Kopiejewski, Christelle L'Ebraly,