日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Design, Synthesis, and Pharmacokinetic Profiling of Fluorinated Reversible N-Alkyl Carbamate Derivatives of Psilocin for Sub-Hallucinogenic Brain Exposure

氟化可逆N-烷基氨基甲酸酯衍生物(裸盖菇素衍生物)的设计、合成及药代动力学分析,用于亚致幻脑暴露

Banzato, Marco; Colognesi, Martina; Lucatello, Lorena; Comai, Stefano; Pasut, Gianfranco; Capolongo, Francesca; Orian, Laura; Biasutto, Lucia; Signor, Anna; Gabbia, Daniela; Manfredi, Paolo L; De Martin, Sara; Mattarei, Andrea

The Role of Structural Dispersity of Polymer Brushes in Determining the Colloidal Stability of Core-Shell Nanoparticles and Their Interaction with Anti-PEG Antibodies.

聚合物刷的结构分散性在决定核壳纳米粒子的胶体稳定性及其与抗PEG抗体的相互作用中的作用。

Pavón Carlos, Grigoletto Antonella, Kempkes Verena, Eguskiza Ander, Morbidelli Maria, Fiammengo Roberto, Papini Emanuele, Mattarei Andrea, Pasut Gianfranco, Matyjaszewski Krzysztof, Lorandi Francesca, Benetti Edmondo M

Dexamethasone conjugation to an Avidin-Nucleic-Acid-NanoASsembly eliminates the steroid plasma absorption, enhancing selective lung tropism in a murine model of pulmonary fibrosis.

将地塞米松与亲和素-核酸-纳米组装体结合,可消除类固醇的血浆吸收,从而在小鼠肺纤维化模型中增强选择性肺趋向性

Morelli Annalisa, Schiavon Elisa, Violatto Martina Bruna, Moscatiello Giulia Yuri, Salmaso Anita, Passoni Alice, Lanno Alessia, Bernardotto Simone, Stocco Martina, Mattarei Andrea, Bagnati Renzo, Meloni Federica, Bigini Paolo, Morpurgo Margherita

Mitapivat metabolically reprograms human β-thalassemic erythroblasts, increasing their responsiveness to oxidation

Mitapivat 可代谢性地重编程人类β-地中海贫血红细胞,增强其对氧化反应的敏感性。

Siciliano, Angela; D'Alessandro, Angelo; Matte, Alessandro; Bisello, Giovanni; Bertoldi, Mariarita; Dzieciatkowska, Monika; Argabright, Amy; Pozzetto, Richard Huot; Riccardi, Veronica; Mattarei, Andrea; Ongaro, Alberto; Ceolan, Jacopo; Russo, Roberta; Rivadeneyra, Leonardo; Wind-Rotolo, Megan; Iolascon, Achille; Brugnara, Carlo; De Franceschi, Lucia

Mito-Genipin, a Novel Mitochondria-Targeted Genipin Derivative Modulates Oxidative Stress and Inflammation in Macrophages

Mito-Genipin,一种新型线粒体靶向京尼平衍生物,可调节巨噬细胞中的氧化应激和炎症

Angi, Beatrice; Di Molfetta, Daria; Pendin, Diana; Antoniazzi, Giuseppe; Flora, Carlo Alberto; De Leonardis, Francesco; Buono, Martina; Fiermonte, Giuseppe; Szabo, Ildiko; Mattarei, Andrea; Varanita, Tatiana

Letter to the Editor regarding 'Unique pharmacodynamic properties and low abuse liability of the µ-opioid receptor ligand (S)-methadone'

致编辑的信,主题为“μ-阿片受体配体(S)-美沙酮独特的药效学特性和低滥用风险”

Pappagallo, Marco; Kosten, Thomas R; Gorodetzky, Charles W; Vocci, Frank J; Sapienza, Frank L; De Martin, Sara; Comai, Stefano; Mattarei, Andrea; Inturrisi, Charles E; Manfredi, Paolo L

N-methyl-D-aspartate Receptors and Depression: Linking Psychopharmacology, Pathology and Physiology in a Unifying Hypothesis for the Epigenetic Code of Neural Plasticity

N-甲基-D-天冬氨酸受体与抑郁症:将精神药理学、病理学和生理学联系起来,构建神经可塑性表观遗传密码的统一假说

Comai, Stefano; De Martin, Sara; Mattarei, Andrea; Guidetti, Clotilde; Pappagallo, Marco; Folli, Franco; Alimonti, Andrea; Manfredi, Paolo L

Pharmacokinetics, Tolerability, and Safety of Esmethadone in Subjects with Chronic Kidney Disease or Hepatic Impairment

慢性肾病或肝功能损害患者服用艾司美沙酮的药代动力学、耐受性和安全性

Ferri, Nicola; De Martin, Sara; Stuart, James; Traversa, Sergio; Mattarei, Andrea; Comai, Stefano; Folli, Franco; Pappagallo, Marco; Guidetti, Clotilde; Inturrisi, Charles E; Manfredi, Paolo L

The novel uncompetitive NMDA receptor antagonist esmethadone (REL-1017) has no meaningful abuse potential in recreational drug users

新型非竞争性NMDA受体拮抗剂艾司美沙酮(REL-1017)在娱乐性药物使用者中没有明显的滥用潜力。

Shram, Megan J; Henningfield, Jack E; Apseloff, Glen; Gorodetzky, Charles W; De Martin, Sara; Vocci, Frank L; Sapienza, Frank L; Kosten, Thomas R; Huston, Jeff; Buchhalter, August; Ashworth, Judy; Lanier, Ryan; Folli, Franco; Mattarei, Andrea; Guidetti, Clotilde; Comai, Stefano; O'Gorman, Cedric; Traversa, Sergio; Inturrisi, Charles E; Manfredi, Paolo L; Pappagallo, Marco

Esmethadone-HCl (REL-1017): a promising rapid antidepressant

盐酸艾司美沙酮(REL-1017):一种有前景的速效抗抑郁药

Fava, Maurizio; Stahl, Stephen M; De Martin, Sara; Mattarei, Andrea; Bettini, Ezio; Comai, Stefano; Alimonti, Andrea; Bifari, Francesco; Pani, Luca; Folli, Franco; Guidetti, Clotilde; Furlan, Alberto; Sgrignani, Jacopo; Locatelli, Patrizia; Cavalli, Andrea; O'Gorman, Cedric; Traversa, Sergio; Inturrisi, Charles E; Pappagallo, Marco; Manfredi, Paolo L