日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

The PP2A-Integrator-CDK9 axis fine-tunes transcription and can be targeted therapeutically in cancer

PP2A-Integrator-CDK9轴精细调控转录,可作为癌症治疗的靶点。

Stephin J Vervoort,Sarah A Welsh,Jennifer R Devlin,Elisa Barbieri,Deborah A Knight,Sarah Offley,Stefan Bjelosevic,Matteo Costacurta,Izabela Todorovski,Conor J Kearney,Jarrod J Sandow,Zheng Fan,Benjamin Blyth,Victoria McLeod,Joseph H A Vissers,Karolina Pavic,Ben P Martin,Gareth Gregory,Elena Demosthenous,Magnus Zethoven,Isabella Y Kong,Edwin D Hawkins,Simon J Hogg,Madison J Kelly,Andrea Newbold,Kaylene J Simpson,Otto Kauko,Kieran F Harvey,Michael Ohlmeyer,Jukka Westermarck,Nathanael Gray,Alessandro Gardini,Ricky W Johnstone

Targeting histone acetylation dynamics and oncogenic transcription by catalytic P300/CBP inhibition

通过抑制催化性P300/CBP来靶向组蛋白乙酰化动态和致癌转录

Simon J Hogg ,Olga Motorna ,Leonie A Cluse ,Timothy M Johanson ,Hannah D Coughlan ,Ramya Raviram ,Robert M Myers ,Matteo Costacurta ,Izabela Todorovski ,Lizzy Pijpers ,Stefan Bjelosevic ,Tobias Williams ,Shannon N Huskins ,Conor J Kearney ,Jennifer R Devlin ,Zheng Fan ,Jafar S Jabbari ,Ben P Martin ,Mohamed Fareh ,Madison J Kelly ,Daphné Dupéré-Richer ,Jarrod J Sandow ,Breon Feran ,Deborah Knight ,Tiffany Khong ,Andrew Spencer ,Simon J Harrison ,Gareth Gregory ,Vihandha O Wickramasinghe ,Andrew I Webb ,Phillippa C Taberlay ,Kenneth D Bromberg ,Albert Lai ,Anthony T Papenfuss ,Gordon K Smyth ,Rhys S Allan ,Jonathan D Licht ,Dan A Landau ,Omar Abdel-Wahab ,Jake Shortt ,Stephin J Vervoort ,Ricky W Johnstone

Inactivation of CK1α in multiple myeloma empowers drug cytotoxicity by affecting AKT and β-catenin survival signaling pathways

多发性骨髓瘤中 CK1α 失活通过影响 AKT 和 β-catenin 存活信号通路增强药物细胞毒性

Sabrina Manni, Marilena Carrino, Martina Manzoni, Ketty Gianesin, Sara Canovas Nunes, Matteo Costacurta, Laura Quotti Tubi, Paolo Macaccaro, Elisa Taiana, Anna Cabrelle, Gregorio Barilà, Annalisa Martines, Renato Zambello, Laura Bonaldi, Livio Trentin, Antonino Neri, Gianpietro Semenzato, Francesco