日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Erythrosin B is a potent and broad-spectrum orthosteric inhibitor of the flavivirus NS2B-NS3 protease

赤藓红 B 是一种强效、广谱的黄病毒 NS2B-NS3 蛋白酶正构抑制剂

Zhong Li, Srilatha Sakamuru, Ruili Huang, Matthew Brecher, Cheri A Koetzner, Jing Zhang, Haiying Chen, Cheng-Feng Qin, Qing-Yu Zhang, Jia Zhou, Laura D Kramer, Menghang Xia, Hongmin Li

Existing drugs as broad-spectrum and potent inhibitors for Zika virus by targeting NS2B-NS3 interaction

现有药物通过靶向 NS2B-NS3 相互作用作为寨卡病毒的广谱强效抑制剂

Zhong Li, Matthew Brecher, Yong-Qiang Deng, Jing Zhang, Srilatha Sakamuru, Binbin Liu, Ruili Huang, Cheri A Koetzner, Christina A Allen, Susan A Jones, Haiying Chen, Na-Na Zhang, Min Tian, Fengshan Gao, Qishan Lin, Nilesh Banavali, Jia Zhou, Nathan Boles, Menghang Xia, Laura D Kramer, Cheng-Feng Qin

A conformational switch high-throughput screening assay and allosteric inhibition of the flavivirus NS2B-NS3 protease

黄病毒 NS2B-NS3 蛋白酶的构象转换高通量筛选试验和变构抑制

Matthew Brecher, Zhong Li, Binbin Liu, Jing Zhang, Cheri A Koetzner, Adham Alifarag, Susan A Jones, Qishan Lin, Laura D Kramer, Hongmin Li

S-adenosyl-homocysteine is a weakly bound inhibitor for a flaviviral methyltransferase

S-腺苷酸同型半胱氨酸是黄病毒甲基转移酶的弱结合抑制剂

Hui Chen, Bing Zhou, Matthew Brecher, Nilesh Banavali, Susan A Jones, Zhong Li, Jing Zhang, Dilip Nag, Laura D Kramer, Arun K Ghosh, Hongmin Li

Cathepsin cleavage potentiates the Ebola virus glycoprotein to undergo a subsequent fusion-relevant conformational change

组织蛋白酶裂解增强埃博拉病毒糖蛋白发生随后的融合相关构象变化

Matthew Brecher, Kathryn L Schornberg, Sue E Delos, Marnie L Fusco, Erica Ollmann Saphire, Judith M White