Demonstrating In-Cell Target Engagement Using a Pirin Protein Degradation Probe (CCT367766)
使用 Pirin 蛋白降解探针 (CCT367766) 展示细胞内靶标参与
期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/acs.jmedchem.7b01406
Nicola E A Chessum, Swee Y Sharp, John J Caldwell, A Elisa Pasqua, Birgit Wilding, Giampiero Colombano, Ian Collins, Bugra Ozer, Meirion Richards, Martin Rowlands, Mark Stubbs, Rosemary Burke, P Craig McAndrew, Paul A Clarke, Paul Workman, Matthew D Cheeseman, Keith Jones