Achieving In Vivo Target Depletion through the Discovery and Optimization of Benzimidazolone BCL6 Degraders
通过发现和优化苯并咪唑酮 BCL6 降解剂实现体内靶标耗竭
期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/acs.jmedchem.9b02076
Benjamin R Bellenie, Kwai-Ming J Cheung, Ana Varela, Olivier A Pierrat, Gavin W Collie, Gary M Box, Michael D Bright, Sharon Gowan, Angela Hayes, Matthew J Rodrigues, Kartika N Shetty, Michael Carter, Owen A Davis, Alan T Henley, Paolo Innocenti, Louise D Johnson, Manjuan Liu, Selby de Klerk, Yann-V