日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

BET bromodomain inhibition potentiates radiosensitivity in models of H3K27-altered diffuse midline glioma

BET 溴结构域抑制增强了 H3K27 改变的弥漫性中线胶质瘤模型的放射敏感性

Jun Watanabe, Matthew R Clutter, Michael J Gullette, Takahiro Sasaki, Eita Uchida, Savneet Kaur, Yan Mo, Kouki Abe, Yukitomo Ishi, Nozomu Takata, Manabu Natsumeda, Samantha Gadd, Zhiguo Zhang, Oren J Becher, Rintaro Hashizume6

Synergistic PIM kinase and proteasome inhibition as a therapeutic strategy for MYC-overexpressing triple-negative breast cancer

协同抑制PIM激酶和蛋白酶体作为治疗MYC过表达三阴性乳腺癌的策略

Ratika Kunder,Michelle Velyunskiy,Sara F Dunne,Byoung-Kyu Cho,Deepak Kanojia,Lauren Begg,Adrienne M Orriols,Erica Fleming-Trujillo,Pranathi Vadlamani,Alesia Vialichka,Rosemary Bolin,Jessica N Perrino,Diane Roth,Matthew R Clutter,Nicolette A Zielinski-Mozny,Young Ah Goo,Massimo Cristofanilli,Marc L Mendillo,Athanassios Vassilopoulos,Dai Horiuchi

Discovery of a small-molecule inhibitor of the TRIP8b-HCN interaction with efficacy in neurons

发现一种对神经元有效的TRIP8b-HCN相互作用的小分子抑制剂

Ye Han ,Iredia D Iyamu ,Matthew R Clutter ,Rama K Mishra ,Kyle A Lyman ,Chengwen Zhou ,Ioannis Michailidis ,Maya Y Xia ,Horrick Sharma ,Chi-Hao Luan ,Gary E Schiltz ,Dane M Chetkovich

Quantitative and multiplexed chemical-genetic phenotyping in mammalian cells with QMAP-Seq

使用 QMAP-Seq 对哺乳动物细胞进行定量和多重化学遗传表型分析

Sonia Brockway, Geng Wang, Jasen M Jackson, David R Amici, Seesha R Takagishi, Matthew R Clutter, Elizabeth T Bartom, Marc L Mendillo

Discovery of novel Mnk inhibitors using mutation-based induced-fit virtual high-throughput screening

使用基于突变的诱导契合虚拟高通量筛选发现新型 Mnk 抑制剂

Rama K Mishra, Matthew R Clutter, Gavin T Blyth, Ewa M Kosciuczuk, Amy Z Blackburn, Elspeth M Beauchamp, Gary E Schiltz, Leonidas C Platanias

A Chemical Probe Strategy for Interrogating Inhibitor Selectivity Across the MEK Kinase Family

用于探究 MEK 激酶家族抑制剂选择性的化学探针策略

Kristine K Deibler, Rama K Mishra, Matthew R Clutter, Aleksandar Antanasijevic, Raymond Bergan, Michael Caffrey, Karl A Scheidt

Single-cell mass cytometry adapted to measurements of the cell cycle

适用于测量细胞周期的单细胞质谱流式细胞术

Gregory K Behbehani, Sean C Bendall, Matthew R Clutter, Wendy J Fantl, Garry P Nolan

Tyramide signal amplification for analysis of kinase activity by intracellular flow cytometry

酪胺信号放大用于通过细胞内流式细胞术分析激酶活性

Matthew R Clutter, Garrett C Heffner, Peter O Krutzik, Kacey L Sachen, Garry P Nolan